Glycyrrhizina (Licorice Flavonoids & Glycyrrhizic Acid — BGG World)

Glycyrrhiza glabra
Evidence Level
Preliminary
3 Clinical Trials
8 Documented Benefits
1/5 Evidence Score

Glycyrrhizina is BGG World's comprehensive licorice (Glycyrrhiza species) portfolio — BGG has been extracting licorice roots since 1995 with 20+ years controlling the entire production chain. Product range includes: licorice extracts (deglycyrrhizinated/DGL or conventional), glycyrrhizic acid derivatives (Mono Ammonium Glycyrrhizinate/MAG, Enoxolone/18-β-Glycyrrhetinic Acid, Dipotassium Glycyrrhizinate), and licorice flavonoids (Licochalcone A, Glabridin). Licorice has a long history of traditional use. One thing to know before reading further: three of the four references on this page are safety or harm papers, and the fourth is an intravenous drug trial in people with chronic hepatitis C, so not one of them is an oral efficacy study. Licochalcone A and glabridin are used in topical personal care, which is outside the scope of an oral supplement.

Studied Dose No oral dose here is backed by a cited reference; for licorice containing glycyrrhizin, about 10 mg/day of glycyrrhizic acid is a safe intake and 400 mg/day causes adverse effects in most people.
Active Compound Licorice (Glycyrrhiza glabra, G. uralensis) extracts (DGL or conventional); glycyrrhizic acid derivatives (Mono Ammonium Glycyrrhizinate, Enoxolone/18-β-Glycyrrhetinic Acid, Dipotassium Glycyrrhizinate); flavonoids (Licochalcone A, Glabridin).

Benefits

The H. pylori figure is not supported here

A figure of 56% versus 4% on placebo for clearing H. pylori has been quoted for deglycyrrhizinated licorice (DGL), but that study is not among the four references on this page, so the figure is uncited and cannot be checked here. Clearing an infection is also a medical outcome rather than a supplement benefit, and it is not something a supplement may claim. A confirmed H. pylori infection is a matter for your doctor.

Ulcer claims are not supported here

DGL has been described as being as effective as H2 blocker medicines for duodenal ulcer resolution. No reference on this page supports that comparison, and a supplement cannot be presented as an equivalent to prescription medicine for a diagnosed condition. Licorice does have a long traditional use for epigastric discomfort and indigestion, but that describes a tradition rather than a demonstrated effect. Ulcer symptoms need a doctor.

The reflux trial is not cited on this page

A trial of a standardized DGL extract in adults with reflux symptoms is sometimes cited for this ingredient, but it is not among the four references here, so nothing on this page documents it. Gastroesophageal reflux disease is a diagnosed condition and relieving it is not a supplement claim. Persistent heartburn should be looked at by a clinician.

Mucosal effects are mechanistic, not demonstrated

Licorice flavonoids have been described as having anti-inflammatory and antioxidant activity on the gastrointestinal lining. That is laboratory and mechanistic reasoning. No reference on this page measured any digestive outcome in people taking an oral licorice product, so none of it should be read as evidence that a supplement heals tissue or repairs damage caused by medication.

Glabridin is a topical cosmetic ingredient

Glabridin inhibits tyrosinase in laboratory assays, which is why it appears in topical skin-lightening cosmetics applied to the surface of the skin. Nothing on this page shows that swallowing a licorice extract changes skin pigmentation, and this site covers oral supplements only.

Licochalcone A is also a topical ingredient

Licochalcone A is used in leave-on skin care for redness and blemish-prone skin. As with glabridin, that evidence is topical and does not transfer to a capsule taken by mouth. No reference on this page tested either flavonoid taken orally.

Reduced side effect profile via deglycyrrhizination

Deglycyrrhizinated licorice (DGL) has had the glycyrrhizin taken out, so it does not carry the mineralocorticoid effect of native licorice, which produces sodium retention, potassium loss and raised blood pressure. That distinction matters, because the cited work documents real harm from the native compound: systolic blood pressure rose 3.1 to 14.4 mmHg across the doses tested, adverse effects can begin in sensitive people at a regular intake of about 100 mg of glycyrrhizic acid a day, and most people taking 400 mg a day experience them. DGL avoids that mechanism. It does not follow that DGL has a proven benefit, because no oral efficacy study is cited on this page.

Neurological work is in animals only

Licorice flavonoids have been reported to modulate GABA signaling, and liquiritigenin reduced glutamate toxicity in mouse hippocampal neurons. That work is in mice and in isolated cells, and none of it is cited on this page. Animal seizure models describe a disease and cannot support a claim for people, and nothing here shows an effect on human brain function. Treat it as early laboratory background only.

Mechanism of action

1

Mucosal protection via flavonoid anti-inflammatory

Licorice flavonoids have been reported in laboratory work to reduce inflammatory signaling, including NF-κB and COX-2 activity. This is a proposed mechanism for the gastrointestinal lining. It is not tied to any measured outcome in the references on this page.

2

Antimicrobial activity in the laboratory

Licorice-derived flavonoids have shown activity against Helicobacter pylori in laboratory testing. The eradication percentages quoted elsewhere on this page come from a study that is not cited here, so they cannot be verified, and activity in a dish is not evidence that a supplement clears an infection in a person.

3

Tyrosinase inhibition (topical cosmetic use)

Glabridin inhibits tyrosinase, the rate-limiting enzyme in melanin synthesis, in laboratory assays. That is the basis for its use in cosmetics applied to the skin. It is not a mechanism for an oral supplement, and no reference here compares it with any medicine.

4

11β-HSD2 inhibition (native glycyrrhizin)

Native glycyrrhizin (not present in DGL) inhibits 11β-hydroxysteroid dehydrogenase type 2 — the enzyme that inactivates cortisol. Cortisol is then free to act on the mineralocorticoid receptor, which produces sodium and water retention, potassium loss, edema and raised blood pressure. A controlled human study found a linear dose response, with systolic blood pressure rising 3.1 to 14.4 mmHg at intakes of 75 to 540 mg of glycyrrhetinic acid per day over two to four weeks. Deglycyrrhizination removes the compound responsible, and with it this mechanism.

5

GABAergic modulation and neuroprotection

Licorice flavonoid extracts have been reported to modulate GABA signaling, and liquiritigenin reduced glutamate toxicity in mouse hippocampal neurons in cell work. All of this is animal and cell data, none of it is cited on this page, and it says nothing about what an oral licorice supplement does in people.

Clinical trials

1
Uncited: the H. pylori eradication study

This study is not among the four references on this page, and no author, journal, year or PubMed identifier is given for it, so its design and size cannot be checked. It is listed here as uncited.

Not verifiable. The population, the number of participants and the length of the intervention are all unsourced.

The 56% against 4% eradication figure cannot be traced to any reference on this page, so it is reported here only as an unverified claim rather than a supported result. Clearing a bacterial infection is in any case a medical outcome that a supplement may not claim.

2
Uncited: the reflux trial

No reference on this page corresponds to this trial. The phase III label, the design and the 28-day duration are unsourced and cannot be verified.

Given as 200 adults with reflux symptoms, but the figure is unsourced and cannot be confirmed.

Reported as a benefit for reflux symptoms with no citation behind it. Reflux disease is a diagnosed condition and a supplement may not be offered as relief for it. Nothing on this page documents this result.

3
Uncited: licorice flavonoid oil studies

These licorice flavonoid oil studies are not among the references on this page. They also concern a different material from the DGL and glycyrrhizin products described above, so they would not support claims for those even if they were cited.

Given as about 50 people in the knee study and 11 to 17 in the small metabolic studies, all unsourced. Studies of that size are exploratory.

The reported change in trunk muscle mass was a gain of 0.17 kg with the extract against a loss of 0.57 kg on placebo, with standard deviations of about 1 kg, which is wider than the difference between the groups. The AMPK and fat oxidation statements are mechanistic. None of it is cited on this page, and knee osteoarthritis is a diagnosed joint disease that a supplement may not claim to treat.

Side effects and drug interactions

Common Potential side effects

DGL form is generally well tolerated; removing the glycyrrhizin is what removes the blood pressure and potassium risk, though no oral efficacy study for DGL is cited on this page.
Native (non-DGL) licorice at high doses: hypertension, sodium retention, hypokalemia, edema, via 11β-HSD2 inhibition. In a controlled human study systolic blood pressure rose 3.1 to 14.4 mmHg, and as little as 50 g of licorice a day (about 75 mg glycyrrhetinic acid) for two weeks raised it significantly.
Native licorice cardiac arrest case reported in literature (high intake) — adhere to EFSA limit of 100 mg glycyrrhizin/day equivalent.
Pregnancy: avoid. Licorice consumption during pregnancy has been associated with preterm birth.
A long history of use is not a safety record. One of the reviews cited here concludes that daily consumption of licorice is never justified, because its benefits are minor compared with the adverse outcomes of chronic consumption, and it calls for a warning and an upper limit on intake.
Mild GI effects rare with DGL form.
Dose ceilings from the cited work: in the most sensitive people a regular intake of no more than about 100 mg of glycyrrhizic acid a day is enough to produce adverse effects, most people who take 400 mg a day experience them, and about 10 mg a day is described as a safe dose for most healthy adults.

Important Drug interactions

Antihypertensive medications — native licorice causes hypertension via 11β-HSD2 inhibition; DGL form avoids this; use DGL for those on BP medications.
Diuretics (loop, thiazide) — native licorice causes hypokalemia; avoid combining; DGL form is safer.
Digoxin — native licorice hypokalemia increases digoxin toxicity risk; avoid; DGL safer.
Corticosteroids — native licorice prolongs corticosteroid effects via 11β-HSD2 inhibition.
Grapefruit juice — similar 11β-HSD2 inhibition mechanism; possible additive effects.
Anticoagulants (warfarin) — licorice flavonoids may have mild antiplatelet effects.
Pregnancy: avoid. Preterm birth association reported.
Furosemide and other 11β-HSD2 inhibitors — additive effects.

Frequently asked questions about Glycyrrhizina (Licorice Flavonoids & Glycyrrhizic Acid — BGG World)

What is glycyrrhizin used for?

Glycyrrhizin (glycyrrhizic acid) is the main active compound in licorice root, and it is intensely sweet, so it is also used as a flavoring. It is the compound behind licorice's blood pressure and potassium problems, which is why it is stripped out to make deglycyrrhizinated licorice (DGL). The references on this page are about that risk rather than about any oral benefit.

What is glycyrrhizin good for?

The one efficacy study cited on this page is a phase I/II trial of pharmaceutical grade glycyrrhizin given intravenously three times a week for four weeks to people with chronic hepatitis C. Liver enzyme (ALT) levels fell 26% against 6% on placebo, but the virus was not cleared and the effect disappeared once the infusions stopped. That is an intravenous drug study in a diagnosed illness, and it says nothing about what an oral licorice supplement does in a healthy person.

How much glycyrrhizin is safe?

Because glycyrrhizin raises blood pressure and lowers potassium, intake has a real ceiling. European food safety guidance points to an upper limit of about 100 mg a day, and the hazard review cited here reaches a similar place: in the most sensitive people a regular intake of no more than about 100 mg of glycyrrhizic acid a day is enough to produce adverse effects, most people taking 400 mg a day experience them, and about 10 mg a day would be a safe dose for most healthy adults. This is exactly the compound removed to make DGL licorice.

Is glycyrrhizin safe?

In small, occasional amounts it is generally tolerated, but regular or high intake can cause high blood pressure, low potassium, and fluid retention. People with hypertension, heart, or kidney conditions, or who are pregnant, should avoid it.

What is Glycyrrhizina?

Glycyrrhizina is BGG World's comprehensive licorice (Glycyrrhiza species) portfolio — BGG has been extracting licorice roots since 1995 with 20+ years controlling the entire production chain.

What is Glycyrrhizina used for?

Glycyrrhizina is researched primarily for Gut Health. A figure of 56% versus 4% on placebo for clearing H. pylori has been quoted for deglycyrrhizinated licorice (DGL), but that study is not among the four references on this page, so the figure is uncited and cannot be checked here.

What is the recommended dosage of Glycyrrhizina?

The clinically studied dose is No oral dose here is backed by a cited reference; for licorice containing glycyrrhizin, about 10 mg/day of glycyrrhizic acid is a safe intake and 400 mg/day causes adverse effects in most people. Always follow the product label and check with a healthcare provider for personal advice.

Is Glycyrrhizina safe, and does it have side effects?

For most healthy adults, Glycyrrhizina is well tolerated at studied doses. Reported effects can include: DGL form is generally well tolerated; removing the glycyrrhizin is what removes the blood pressure and potassium risk, though no oral efficacy study for DGL is cited on this page. It may also interact with some medications. Glycyrrhizina is not right for everyone, so check with a healthcare provider first if you are pregnant or breastfeeding, have a medical condition, or take prescription medication.

Does Glycyrrhizina interact with any medications?

Possible interactions include: Antihypertensive medications — native licorice causes hypertension via 11β-HSD2 inhibition; DGL form avoids this; use DGL for those on BP medications. Diuretics (loop, thiazide) — native licorice causes hypokalemia; avoid combining; DGL form is safer. If you take prescription medication, check with a pharmacist or doctor before using it.

How strong is the scientific evidence for Glycyrrhizina?

NutraSmarts rates the evidence for Glycyrrhizina as Preliminary (1 out of 5). It is backed by 3 clinical trials and 4 cited references summarized on this page. A higher rating reflects more, larger, and better-designed human studies.

References(4 citations)

Evidence ratings on NutraSmarts are based on the totality of human clinical research, with emphasis on randomized controlled trials, meta-analyses, and systematic reviews. The references below directly support claims made throughout this page.

  1. Omar HR, Komarova I, El-Ghonemi M, Fathy A, Rashad R, Abdelmalak HD, Yerramadha MR, Ali Y, et al. Licorice abuse: time to send a warning message Ther Adv Endocrinol Metab. 2012;3(4):125-38. doi: 10.1177/2042018812454322.PubMedUsed to support: Leads the safety angle: comprehensive review documenting that glycyrrhizin inhibits 11-beta-HSD2, causing pseudohyperaldosteronism - sodium/water retention, hypertension, hypokalemia, edema and arrhythmia risk with sustained or high intake. Honesty: this is a well-documented real harm; deglycyrrhizinated licorice (DGL) avoids it.
  2. Sigurjonsdottir HA, Franzson L, Manhem K, Ragnarsson J, Sigurdsson G, Wallerstedt S Liquorice-induced rise in blood pressure: a linear dose-response relationship J Hum Hypertens. 2001;15(8):549-52. doi: 10.1038/sj.jhh.1001215.PubMedUsed to support: Quantifies the hypertension harm: a controlled human study showing licorice (glycyrrhetinic acid) raises systolic blood pressure in a linear, dose-dependent way. Honesty: confirms even moderate sustained intake can elevate BP, reinforcing strict dose limits and caution in hypertensives.
  3. van Rossum TG, Vulto AG, Hop WC, Brouwer JT, Niesters HG, Schalm SW Intravenous glycyrrhizin for the treatment of chronic hepatitis C: a double-blind, randomized, placebo-controlled phase I/II trial J Gastroenterol Hepatol. 1999;14(11):1093-9. doi: 10.1046/j.1440-1746.1999.02008.x.PubMedUsed to support: Backs glycyrrhizin's recognized therapeutic use: intravenous glycyrrhizin (the active principle of Stronger Neo-Minophagen C) lowered serum ALT/aminotransferases in chronic hepatitis C. Honesty: the benefit is on liver-enzyme markers using the IV form; it does not eradicate the virus, and oral/high-dose use carries the mineralocorticoid harms noted above.
  4. Stormer FC, Reistad R, Alexander J Glycyrrhizic acid in liquorice--evaluation of health hazard Food Chem Toxicol. 1993;31(4):303-12. doi: 10.1016/0278-6915(93)90080-i.PubMedUsed to support: Reinforces the safety/dose-limit angle: a health-hazard evaluation of glycyrrhizic acid establishing tolerable-intake estimates and documenting that habitual intake can cause pseudohyperaldosteronism (hypertension, hypokalemia). Honesty: frames glycyrrhizin as a compound with a real ceiling on safe intake, not a benign botanical.