Venetron® (Rafuma / Apocynum venetum Leaf Extract)

Apocynum venetum
Evidence Level
Limited
1 Clinical Trial
3 Documented Benefits
2/5 Evidence Score

Venetron® (Tokiwa Phytochemical) is a standardized extract of Apocynum venetum (Luobuma/Rafuma) leaves — a traditional Chinese herbal medicine used for over 2,000 years for hypertension, anxiety, and insomnia. It is standardized for two flavonoids, hyperoside and isoquercitrin. Laboratory and animal work suggests these compounds act on serotonin signalling, but that has not been shown to produce a mood or anxiety effect in people. The only human study cited on this page measured sleep, none of the cited research tested blood pressure, and nothing cited compares this extract with a prescription antidepressant or sedative.

Studied Dose 50 mg/day.
Active Compound Standardized Apocynum venetum leaf extract, standardized for hyperoside and isoquercitrin (quercetin glycosides); 50 mg/day.

Benefits

Mood: animal research only, no human data

No human study cited on this page measured mood. This claim rests entirely on a 2013 rodent study in which flavonoids from Apocynum venetum leaves changed brain monoamine levels and produced antidepressant-like behaviour in animals. There are no depression scores from people, no placebo comparison in people, and no head-to-head comparison with an antidepressant medicine. Depression is a medical condition; if you are struggling with low mood, speak to a doctor rather than relying on a supplement.

Calming use is traditional, not tested here

None of the studies cited on this page measured anxiety or stress in people. The plant has a long history of use as a calming tea in China, and a review article describes that tradition, but traditional use is not the same as tested. The receptor effects described for hyperoside and isoquercitrin come from laboratory work, not from people taking the supplement.

Sleep: more deep sleep in one small brain-wave study

This is the one area with any human data. In a small 2015 study that recorded sleep with EEG, 50 mg of Apocynum venetum leaf extract taken on its own increased non-REM (deeper) sleep time by 7.6%. It did not shorten the time taken to fall asleep; GABA on its own did that, by about 5.3 minutes, and combining the two was no better than either alone. More non-REM time on a sleep trace is a laboratory measurement, not proof that people woke up feeling more rested, and a single small study is a thin basis for a sleep claim.

Mechanism of action

1

What the flavonoids do in the lab, and what that does not prove

In laboratory and animal work, hyperoside and isoquercitrin appear to affect serotonin signalling, and a rodent study reported changes in brain serotonin, dopamine and noradrenaline. That is a plausible idea about how the extract might work, not something measured in people. It does not make the extract equivalent to fluoxetine, sertraline or any other prescription medicine, and no human study cited here measured mood, anxiety or brain chemistry.

Clinical trials

1
Apocynum venetum leaf extract, GABA and sleep EEG (2015, PMID 26052150)

A small human study that recorded sleep with EEG. It compared GABA on its own, Apocynum venetum leaf extract on its own at 50 mg, and the two combined.

A small group of adults. Sleep was measured on a brain-wave recording; mood and anxiety were not assessed.

The leaf extract alone at 50 mg increased non-REM (deeper) sleep time by 7.6%. GABA alone shortened the time to fall asleep by 5.3 minutes. The combination gave 4.3 minutes and 5.1% more non-REM sleep, so it was not better than either ingredient on its own. No depression, anxiety or mood outcome was measured, and the study reports sleep-trace measurements rather than how rested people said they felt. It is a single small study.

Side effects and drug interactions

Common Potential side effects

Appears well tolerated at 50 mg/day, though the human evidence is limited to one small short study
Mild GI effects possible — take with food
Effects on serotonin have only been seen in laboratory and animal work, so any serotonin syndrome concern alongside other serotonin-raising medicines is theoretical rather than reported

Important Drug interactions

SSRIs and SNRIs: no interaction has actually been reported with this extract, but because lab work suggests an effect on serotonin, check with your doctor before combining
MAO inhibitors: no cases have been reported with this extract, but given the theoretical serotonin effect, do not combine without medical advice
Benzodiazepines: no interaction has been studied; any added drowsiness is theoretical, so tell your doctor if you take both

Frequently asked questions about Venetron® (Rafuma / Apocynum venetum Leaf Extract)

What is Venetron?

Venetron® (Tokiwa Phytochemical) is a standardized extract of Apocynum venetum (Luobuma/Rafuma) leaves — a traditional Chinese herbal medicine used for over 2,000 years for hypertension, anxiety, and insomnia. It is standardized for two flavonoids, hyperoside and isoquercitrin.

What is Venetron used for?

Venetron is researched primarily for Sleep Health. No human study cited on this page measured mood. This claim rests entirely on a 2013 rodent study in which flavonoids from Apocynum venetum leaves changed brain monoamine levels and produced antidepressant-like behaviour in animals.

What is the recommended dosage of Venetron?

The clinically studied dose is 50 mg/day. Always follow the product label and check with a healthcare provider for personal advice.

Is Venetron safe, and does it have side effects?

For most healthy adults, Venetron is well tolerated at studied doses. Reported effects can include: Appears well tolerated at 50 mg/day, though the human evidence is limited to one small short study Mild GI effects possible — take with food It may also interact with some medications. Venetron is not right for everyone, so check with a healthcare provider first if you are pregnant or breastfeeding, have a medical condition, or take prescription medication.

Does Venetron interact with any medications?

Possible interactions include: SSRIs and SNRIs: no interaction has actually been reported with this extract, but because lab work suggests an effect on serotonin, check with your doctor before combining MAO inhibitors: no cases have been reported with this extract, but given the theoretical serotonin effect, d… If you take prescription medication, check with a pharmacist or doctor before using it.

How strong is the scientific evidence for Venetron?

NutraSmarts rates the evidence for Venetron as Limited (2 out of 5). It is backed by 1 clinical trial and 4 cited references summarized on this page. A higher rating reflects more, larger, and better-designed human studies.

References(4 citations)

Evidence ratings on NutraSmarts are based on the totality of human clinical research, with emphasis on randomized controlled trials, meta-analyses, and systematic reviews. The references below directly support claims made throughout this page.

  1. Kim D, Choi G, Kim S, Kim J, Oh D, Jin T, Yang J, Cho S Sleep-promoting effects and potential mechanisms of Apocynum venetum leaf extract (VENETRON®): Effects of acute and chronic treatment on the sleep-wake profiles in mice. J Ethnopharmacol. 2025;350:120008. doi: 10.1016/j.jep.2025.120008.PubMedUsed to support: A mouse study. It used the Venetron brand extract and tracked sleep-wake patterns after single and repeated doses. Naming the brand does not make it human evidence, so it cannot support a sleep claim for people.
  2. Yamatsu A, Yamashita Y, Maru I, Yang J, Tatsuzaki J, Kim M The Improvement of Sleep by Oral Intake of GABA and Apocynum venetum Leaf Extract. J Nutr Sci Vitaminol (Tokyo). 2015;61(2):182-7. doi: 10.3177/jnsv.61.182.PubMedUsed to support: The only human study cited on this page. Sleep was recorded by EEG, and the study did include an arm taking 50 mg of Apocynum venetum leaf extract on its own, which increased non-REM (deeper) sleep time by 7.6%. GABA alone shortened the time to fall asleep by 5.3 minutes; the two together gave 4.3 minutes and 5.1% more non-REM sleep, so the combination was no better than either ingredient alone. It is a small study of sleep traces, not of how rested people reported feeling.
  3. Zheng M, Fan Y, Shi D, Liu C Antidepressant-like effect of flavonoids extracted from Apocynum venetum leaves on brain monoamine levels and dopaminergic system. J Ethnopharmacol. 2013;147(1):108-13. doi: 10.1016/j.jep.2013.02.015.PubMedUsed to support: An animal study. Flavonoids from Apocynum venetum leaves changed brain monoamine levels and produced antidepressant-like behaviour in rodents. An animal antidepressant model is not evidence of a mood benefit in people, and no human study cited here measured mood at all.
  4. Xie W, Zhang X, Wang T, Hu J Botany, traditional uses, phytochemistry and pharmacology of Apocynum venetum L. (Luobuma): A review. J Ethnopharmacol. 2012;141(1):1-8. doi: 10.1016/j.jep.2012.02.003.PubMedUsed to support: A review article, not a study. It describes the plant's traditional use for high blood pressure, anxiety and sleeplessness and summarises the chemistry of hyperoside and isoquercitrin. A review collects other people's work; it does not test anything in people and cannot support a benefit claim on its own.