Raspberry Ketone (Rheosmin)

Evidence Level
Preliminary
4 Clinical Trials
5 Documented Benefits
1/5 Evidence Score

Raspberry ketone is the compound that gives red raspberries their smell. The fruit holds only a few milligrams per kilogram, and in the US the chemical is listed as a synthetic flavoring allowed in the minimum amount needed for taste, yet weight-loss supplements recommend 100 to 1,400 mg a day. The fat-burning story comes from mouse and cell studies, where much of the effect traced back to animals simply eating less. No published trial has tested raspberry ketone on its own in people: the two human trials used capsules that also contained caffeine, capsaicin and bitter orange, so they cannot say what the ketone itself did. Safety data at supplement doses are thin, and high doses were toxic in mice.

Studied Dose Not tested alone in humans; products recommend 100-1,400 mg/day
Active Compound 4-(4-Hydroxyphenyl)-2-butanone (raspberry ketone, rheosmin)

Benefits

Weight loss support tested only in stimulant blends

In two randomized trials, overweight adults on a calorie-restricted diet and exercise program took capsules combining raspberry ketone with caffeine, capsaicin, garlic and bitter orange. One reported more weight and fat loss than placebo among the people who finished; in the other, both groups lost weight. With known stimulants in the mix, neither trial can credit the ketone.

Appetite and body fat changes in mice follow reduced food intake

Mice given raspberry ketone ate less and gained less weight. In a study that fed a comparison group the same reduced amount of food, the authors concluded the ketone offered limited fat-loss benefit beyond eating less. In another, doses that reliably cut intake also caused organ changes and deaths. No study has measured appetite in people taking it alone.

Lipolysis and adiponectin effects seen in fat cells

In isolated rat fat cells, raspberry ketone boosted norepinephrine-triggered fat breakdown, and in cultured mouse fat cells it raised fatty acid burning and adiponectin release. These are laboratory results. In the two human blend trials, adiponectin did not change in one and rose in the other, which says little about the ketone itself.

Raspberry aroma compound, not a raspberry extract

Raspberry ketone is a flavor molecule. Raspberries contain up to about 4.3 mg per kilogram, so a single 100 mg serving would take more than 20 kg of fruit. In the US it is listed as a synthetic flavoring substance permitted in the minimum amount needed for flavor, and that listing does not address supplement-level daily intake.

Safety at supplement doses is not established

Formal toxicity data come only from short-term rodent studies, and high doses killed mice in two of them. Danish food safety scientists calculated that the lowest labeled dose, 100 mg, is 56 times the threshold of toxicological concern for its chemical class, with a safety margin of only 12 at 1,400 mg. UK regulators have regarded the pure compound as a novel food that needs authorization.

Mechanism of action

1

Hormone-sensitive lipase and norepinephrine-driven lipolysis

In rat fat cells, raspberry ketone increased the fat breakdown triggered by norepinephrine and moved hormone-sensitive lipase from the cell interior onto lipid droplets, where the enzyme acts. The finding comes from isolated animal cells and has not been measured in human fat tissue.

2

Adiponectin and fatty acid oxidation in cultured adipocytes

At 10 micromolar in 3T3-L1 mouse fat cells, raspberry ketone increased lipolysis, fatty acid oxidation and adiponectin expression and secretion while reducing lipid accumulation. Whether oral doses in people produce tissue concentrations like these is unknown, because human pharmacokinetic data are lacking.

3

Reduced food intake as the main driver in animals

In mice, lower weight gain on raspberry ketone went with eating less. A 200 mg/kg oral dose cut 24-hour intake by 24% in males and 640 mg/kg cut it by 49-77%, without signs of nausea-type behavior, but that higher single dose killed 6 of 14 male mice within two days.

4

Structural kinship with synephrine and capsaicin

Raspberry ketone resembles synephrine and capsaicin in structure, a likeness that prompted the first rodent obesity study. Clinicians reporting coronary artery spasm after a first dose raised the possibility of an adrenaline-like sympathetic effect; that link remains a hypothesis.

Clinical trials

1
Prograde Metabolism Blend with Diet and Exercise
PubMed

Randomized, double-blind, placebo-controlled 8-week trial of a multi-ingredient product containing raspberry ketone, caffeine, capsaicin, garlic, ginger and Citrus aurantium, sponsored by Ultimate Wellness Systems (Lopez HL, Ziegenfuss TN, Hofheins JE, Habowski SM, Arent SM, Weir JP, Ferrando AA 2013, J Int Soc Sports Nutr 10(1):22, PMID 23601452). It did not test raspberry ketone alone.

70 obese but otherwise healthy adults on a calorie-restricted diet with exercise training; 45 completed and were analyzed (27 on the blend, 18 on placebo).

Among completers, body weight fell 2.0% on the blend versus 0.5% on placebo and fat mass 7.8% versus 2.8%, with larger waist and hip reductions. Heart rate, blood pressure and blood chemistries did not differ between groups. More than a third of participants dropped out, the capsules contained caffeine and bitter orange, and two authors reported research funding from or consulting for supplement companies including the sponsor, so the result cannot be credited to raspberry ketone.

2
Multi-Ingredient Blend in Overweight Adults
PubMed

Randomized, double-blind, placebo-controlled 8-week trial of 4 capsules a day of a supplement containing raspberry ketone, capsaicin, caffeine, garlic and Citrus aurantium, by the same research group (Arent SM, Walker AJ, Pellegrino JK, Sanders DJ, McFadden BA, Ziegenfuss TN, Lopez HL 2018, J Am Coll Nutr 37(2):111-120, PMID 29111889). It did not test raspberry ketone alone.

36 overweight men and women, 18 per group, on calorie restriction with supervised exercise three times a week.

Weight, fat mass and body fat percentage fell in both groups, and the abstract does not report a supplement advantage for those outcomes. Group differences were limited to a lean mass gain in men, a larger hip girth reduction in women, lower leptin and higher adiponectin. Any contribution from raspberry ketone cannot be separated from the stimulants in the blend.

3
Pair-Fed Mouse Study (Preclinical)
PubMed

Animal study comparing high-fat diets containing 0.25% or 1.74% raspberry ketone with a control diet and a pair-fed group (Cotten BM, Diamond SA, Banh T, et al. 2017, Food Funct 8(4):1512-1518, PMID 28378858). No humans were studied.

C57BL/6 mice fed a high-fat diet for two weeks, then five weeks on the test diets.

Both doses reduced food intake and body weight compared with control. The low dose did not change liver fat compared with pair-fed mice eating the same amount, and plasma adiponectin was unchanged. The high dose, which had no matched pair-fed group, gave the lowest liver fat and less inguinal fat relative to body weight but a heavier liver. The authors concluded raspberry ketone has limited benefit for fat loss beyond reducing energy intake.

4
Feeding Suppression and Toxicity in Mice (Preclinical)
PubMed

Animal study of single oral doses of 64 to 640 mg/kg raspberry ketone (Hao L, Kshatriya D, Li X, et al. 2020, Food Chem Toxicol 143:111512, PMID 32565406). No humans were studied.

Male and female C57BL/6J mice.

Cumulative 24-hour food intake fell 24% at 200 mg/kg in males and 49-77% at 640 mg/kg. A single 640 mg/kg dose killed 6 of 14 male mice within two days, with white fat atrophy, spleen abnormalities, thymus shrinkage and lower white blood cell counts. The authors concluded that doses which reliably suppress feeding are associated with pathological changes.

Side effects and drug interactions

Common Potential side effects

No human safety study of raspberry ketone alone exists; labeled doses of 100-1,400 mg/day have not been shown to be safe.
A published case describes a 47-year-old woman with a racing heart, blood pressure of 197/130, sweating and diarrhea two hours after her first dose, followed by repeated coronary artery spasm; she had other conditions and causation is unproven.
In mice, a single 640 mg/kg oral dose killed 6 of 14 males and caused fat tissue wasting and immune cell changes; in another study, 10 days at 330 or 500 mg/kg killed half or more of obese mice and raised the liver enzyme ALT.
Computer toxicity models flagged possible effects on the heart and on reproduction or development; avoid during pregnancy and breastfeeding.
Skin contact is a known cause of occupational skin depigmentation, and human liver enzymes in laboratory tests convert it to rhododendrol, a related depigmenting agent; the effect of oral use on skin pigment is unknown.
Many products are blends with caffeine, bitter orange (synephrine) or capsaicin; check the full label for total stimulant content.

Important Drug interactions

No human interaction studies exist for raspberry ketone; the precautions below rest on its proposed adrenergic action, one case report and animal or laboratory data.
Caffeine, synephrine (bitter orange), yohimbine and other stimulant weight-loss ingredients: possible additive effects on heart rate and blood pressure.
ADHD stimulant medicines and decongestants such as pseudoephedrine: the same additive cardiovascular concern.
Blood pressure and heart rhythm medicines: a case of severe hypertension and coronary spasm after a first dose warrants prescriber advice before combining.
Diabetes medicines: in mice, raspberry ketone raised blood glucose in some experiments and lowered it in others; monitor glucose if combining.
Drugs cleared by glucuronidation (UGT enzymes): a laboratory screen found only weak inhibition, so this route of interaction looks unlikely.

Frequently asked questions about Raspberry Ketone (Rheosmin)

What is Raspberry Ketone?

Raspberry ketone is the compound that gives red raspberries their smell. The fruit holds only a few milligrams per kilogram, and in the US the chemical is listed as a synthetic flavoring allowed in the minimum amount needed for taste, yet weight-loss supplements recommend 100 to 1,400 mg a day.

What is Raspberry Ketone used for?

Raspberry Ketone is researched primarily for Weight Management. In two randomized trials, overweight adults on a calorie-restricted diet and exercise program took capsules combining raspberry ketone with caffeine, capsaicin, garlic and bitter orange.

What is the recommended dosage of Raspberry Ketone?

The clinically studied dose is Not tested alone in humans; products recommend 100-1,400 mg/day Always follow the product label and check with a healthcare provider for personal advice.

Is Raspberry Ketone safe, and does it have side effects?

For most healthy adults, Raspberry Ketone is well tolerated at studied doses. Reported effects can include: No human safety study of raspberry ketone alone exists; labeled doses of 100-1,400 mg/day have not been shown to be safe. A published case describes a 47-year-old woman with a racing heart, blood pressure of 197/130, sweating and diarrhea two hours after her first dose, followed… It may also interact with some medications. Raspberry Ketone is not right for everyone, so check with a healthcare provider first if you are pregnant or breastfeeding, have a medical condition, or take prescription medication.

Does Raspberry Ketone interact with any medications?

Possible interactions include: No human interaction studies exist for raspberry ketone; the precautions below rest on its proposed adrenergic action, one case report and animal or laboratory data. If you take prescription medication, check with a pharmacist or doctor before using it.

How strong is the scientific evidence for Raspberry Ketone?

NutraSmarts rates the evidence for Raspberry Ketone as Preliminary (1 out of 5). It is backed by 4 clinical trials and 8 cited references summarized on this page. A higher rating reflects more, larger, and better-designed human studies.

References(8 citations)

Evidence ratings on NutraSmarts are based on the totality of human clinical research, with emphasis on randomized controlled trials, meta-analyses, and systematic reviews. The references below directly support claims made throughout this page.

  1. Lopez HL, Ziegenfuss TN, Hofheins JE, Habowski SM, Arent SM, Weir JP, Ferrando AA. Eight weeks of supplementation with a multi-ingredient weight loss product enhances body composition, reduces hip and waist girth, and increases energy levels in overweight men and women. J Int Soc Sports Nutr. 2013;10(1):22..PubMedUsed to support: The main human trial cited for raspberry ketone, which actually tested a blend with caffeine, capsaicin, garlic, ginger and Citrus aurantium. Among the 45 of 70 participants who completed 8 weeks of diet and exercise, weight and fat mass fell more on the blend than on placebo. Sponsored by Ultimate Wellness Systems; two authors reported research funding from or consulting for supplement companies including the sponsor. It did not test raspberry ketone alone.
  2. Arent SM, Walker AJ, Pellegrino JK, Sanders DJ, McFadden BA, Ziegenfuss TN, Lopez HL. The Combined Effects of Exercise, Diet, and a Multi-Ingredient Dietary Supplement on Body Composition and Adipokine Changes in Overweight Adults. J Am Coll Nutr. 2018;37(2):111-120..PubMedUsed to support: A second 8-week blend trial from the same research group in 36 overweight adults: weight, fat mass and body fat fell in both the supplement and placebo groups, with group differences limited to lean mass in men, hip girth in women, leptin and adiponectin. It did not test raspberry ketone alone.
  3. Morimoto C, Satoh Y, Hara M, Inoue S, Tsujita T, Okuda H. Anti-obese action of raspberry ketone. Life Sci. 2005;77(2):194-204..PubMedUsed to support: The original rodent study behind the weight-loss marketing: raspberry ketone at 0.5-2% of a high-fat diet limited weight, liver and visceral fat gain in mice and increased norepinephrine-induced lipolysis with translocation of hormone-sensitive lipase in rat fat cells. It also notes the structural similarity to capsaicin and synephrine. Animal and cell data only.
  4. Park KS. Raspberry ketone increases both lipolysis and fatty acid oxidation in 3T3-L1 adipocytes. Planta Med. 2010;76(15):1654-8..PubMedUsed to support: Cell-culture study in which 10 micromolar raspberry ketone increased lipolysis, fatty acid oxidation and adiponectin expression and secretion and suppressed lipid accumulation in 3T3-L1 adipocytes. Supports the mechanism section; no animals or humans were studied.
  5. Cotten BM, Diamond SA, Banh T, Hsiao YH, Cole RM, Li J, Simons CT, Bruno RS, Belury MA, Vodovotz Y. Raspberry ketone fails to reduce adiposity beyond decreasing food intake in C57BL/6 mice fed a high-fat diet. Food Funct. 2017;8(4):1512-1518..PubMedUsed to support: An independent pair-fed mouse study concluding that raspberry ketone has limited benefit for fat loss beyond reducing food intake, with plasma adiponectin unchanged. The source of the point that the rodent weight effect largely tracks eating less.
  6. Hao L, Kshatriya D, Li X, Badrinath A, Szmacinski Z, Goedken MJ, Polunas M, Bello NT. Acute feeding suppression and toxicity of raspberry ketone [4-(4-hydroxyphenyl)-2-butanone] in mice. Food Chem Toxicol. 2020;143:111512..PubMedUsed to support: Mouse study showing dose-dependent feeding suppression (24% at 200 mg/kg in males, 49-77% at 640 mg/kg), with a single 640 mg/kg dose killing 6 of 14 male mice and causing white fat atrophy, spleen and thymus changes and lower white blood cell counts. Supports the appetite mechanism and the safety warnings.
  7. Bredsdorff L, Wedebye EB, Nikolov NG, Hallas-Møller T, Pilegaard K. Raspberry ketone in food supplements--High intake, few toxicity data--A cause for safety concern? Regul Toxicol Pharmacol. 2015;73(1):196-200..PubMedUsed to support: Risk assessment from the Technical University of Denmark: supplements recommend 100-1,400 mg/day against natural raspberry content of up to 4.3 mg/kg; 100 mg is 56 times the threshold of toxicological concern; the margin of safety is 165 at 100 mg and 12 at 1,400 mg; QSAR models flagged possible cardiotoxic and reproductive or developmental effects; the UK regarded the pure compound as a novel food requiring authorisation.
  8. Khattar A, Beeton I. Coronary vasospasm and raspberry ketones weight-loss supplement: Is there a connection? Anatol J Cardiol. 2020;24(3):205-208..PubMedUsed to support: Case report of a 47-year-old woman who developed tachycardia, blood pressure of 197/130, sweating and diarrhea about two hours after her first raspberry ketone dose, followed by recurrent episodes highly suggestive of coronary vasospasm with unobstructed coronary arteries. The authors considered raspberry ketone the likely main contributor through a sympathetic mechanism, but no rechallenge was done and she had other active conditions, including anemia requiring transfusion and pulmonary emboli.