Melostacio® (Mango Leaf Extract)

Mangifera indica
Evidence Level
Limited
1 Clinical Trial
3 Documented Benefits
2/5 Evidence Score

Melostacio® (Botanic Healthcare) is a standardized mango leaf (Mangifera indica) extract providing a concentrated source of mangiferin, a plant compound studied for antioxidant and metabolic effects. Mango leaves have a long history of traditional use. Human evidence is limited: the main trial was a 12 week study of 150 mg/day of generic mangiferin (not the Melostacio brand) in 97 overweight adults who had already been diagnosed with high blood fats. It lowered triglycerides and free fatty acids and raised HDL cholesterol, but showed no difference versus placebo in total cholesterol, LDL, fasting blood sugar or insulin. The alpha-glucosidase and AMPK effects come from laboratory and animal work, not from human trials.

Studied Dose The only human trial used 150 mg/day of mangiferin (generic, not Melostacio) for 12 weeks. Doses of 100 to 300 mg/day are commonly listed for standardized mango leaf extracts, but no published trial has tested Melostacio itself.
Active Compound Mangiferin (1,3,6,7-tetrahydroxyxanthone-C2-β-D-glucoside) — Melostacio® by Botanic Healthcare; standardized Mangifera indica leaf extract; primary bioactive mangiferin ≥40%

Benefits

Carbohydrate and glucose handling: laboratory and animal evidence only

In test tube and animal studies, mangiferin slows carbohydrate-digesting enzymes (alpha-glucosidase and alpha-amylase) and switches on AMPK, a cellular energy sensor, in muscle and liver cells. An animal meta-analysis of 19 preclinical studies found lower blood glucose in animals. Human data do not match this yet: in the one 12 week randomized trial (97 overweight adults with high blood fats, 150 mg/day mangiferin), there was no difference between mangiferin and placebo in fasting blood sugar or insulin, although a calculated insulin resistance index did improve. It is not a substitute for diabetes medication.

Anti-inflammatory and antioxidant protection

In laboratory studies mangiferin scavenges free radicals and dampens the NF-kB inflammatory pathway, lowering signaling molecules such as TNF-alpha, IL-6 and IL-1 beta. This comes from a narrative review of laboratory and animal work rather than from human trials. The one human trial cited here reported lipid, glucose and insulin outcomes, not inflammatory markers, so it is unknown whether these effects happen in people at supplement doses.

Lipid profile and cardiovascular support

The human evidence here is real but narrow. In a 12 week double-blind randomized trial of 150 mg/day mangiferin in 97 overweight adults already diagnosed with high blood fats, triglycerides and free fatty acids fell and HDL cholesterol rose compared with placebo. In that same trial there was no difference in total cholesterol or LDL cholesterol, so a claim about lowering cholesterol or LDL is not supported. The trial tested generic mangiferin rather than Melostacio, and it was run in people with a diagnosed lipid condition, so the results may not apply to healthy consumers.

Mechanism of action

1

AMPK activation and alpha-glucosidase inhibition (laboratory and animal studies)

In cell and animal studies, mangiferin activates AMP-activated protein kinase (AMPK), which moves the glucose transporter GLUT4 to cell membranes and increases glucose uptake, and it also blocks the intestinal enzyme alpha-glucosidase, which slows carbohydrate digestion. This is a proposed mechanism, not a proven human effect: the single human trial cited on this page found no change in fasting blood sugar or insulin compared with placebo.

Clinical trials

1
Mangiferin in overweight adults with high blood fats: 12 week randomized trial
PubMed

Randomized, double-blind, placebo-controlled trial of 150 mg/day of generic mangiferin (not the Melostacio brand) for 12 weeks in 97 overweight adults who had been diagnosed with high blood fats. Main outcomes were blood lipids, blood sugar and insulin. (Na et al. 2015, Sci Rep, PMID 25989216)

97 overweight adults with diagnosed hyperlipidemia (high triglycerides or high total cholesterol). Not healthy consumers, and not people with type 2 diabetes.

Triglycerides and free fatty acids dropped and HDL cholesterol rose compared with placebo, and a calculated insulin resistance index improved. There was no difference between the groups in total cholesterol, LDL cholesterol, fasting blood sugar or insulin. Limitations: this is a single trial, it used generic mangiferin rather than Melostacio, and it was run in people already diagnosed with a lipid condition, so the results may not carry over to healthy people or to other mango leaf extracts.

Side effects and drug interactions

Common Potential side effects

Human safety data are limited to one 12 week trial; longer term safety has not been studied
Mild GI effects possible — take with food
Mango allergy (rare) — avoid if known mango allergy (cross-reactivity with leaves)

Important Drug interactions

Antidiabetic medications (insulin, metformin, sulfonylureas): the human trial found no blood sugar change, but animal studies show glucose lowering, so monitor blood glucose and speak with your doctor before combining
Anticoagulants — mangiferin has mild antiplatelet activity; monitor if on blood thinners
Laboratory studies suggest mangiferin can inhibit the CYP2C8 liver enzyme. This has not been tested in people, so check with a pharmacist if you take a CYP2C8-sensitive medication

Frequently asked questions about Melostacio® (Mango Leaf Extract)

What is Melostacio?

Melostacio® (Botanic Healthcare) is a standardized mango leaf (Mangifera indica) extract providing a concentrated source of mangiferin, a plant compound studied for antioxidant and metabolic effects. Mango leaves have a long history of traditional use.

What is Melostacio used for?

Melostacio is researched primarily for Metabolic Health and Antioxidant. In test tube and animal studies, mangiferin slows carbohydrate-digesting enzymes (alpha-glucosidase and alpha-amylase) and switches on AMPK, a cellular energy sensor, in muscle and liver cells.

What is the recommended dosage of Melostacio?

The clinically studied dose is The only human trial used 150 mg/day of mangiferin (generic, not Melostacio) for 12 weeks. Doses of 100 to 300 mg/day are commonly listed for standardized mango leaf extracts, but no published trial has tested Melostacio itself. Always follow the product label and check with a healthcare provider for personal advice.

Is Melostacio safe, and does it have side effects?

For most healthy adults, Melostacio is well tolerated at studied doses. Reported effects can include: Human safety data are limited to one 12 week trial; longer term safety has not been studied Mild GI effects possible — take with food It may also interact with some medications. Melostacio is not right for everyone, so check with a healthcare provider first if you are pregnant or breastfeeding, have a medical condition, or take prescription medication.

Does Melostacio interact with any medications?

Possible interactions include: Antidiabetic medications (insulin, metformin, sulfonylureas): the human trial found no blood sugar change, but animal studies show glucose lowering, so monitor blood glucose and speak with your doctor before combining Anticoagulants — mangiferin has mild antiplatelet activity; mo… If you take prescription medication, check with a pharmacist or doctor before using it.

How strong is the scientific evidence for Melostacio?

NutraSmarts rates the evidence for Melostacio as Limited (2 out of 5). It is backed by 1 clinical trial and 3 cited references summarized on this page. A higher rating reflects more, larger, and better-designed human studies.

References(3 citations)

Evidence ratings on NutraSmarts are based on the totality of human clinical research, with emphasis on randomized controlled trials, meta-analyses, and systematic reviews. The references below directly support claims made throughout this page.

  1. Na L, Zhang Q, Jiang S, Du S, Zhang W, Li Y, Sun C, Niu Y Mangiferin supplementation improves serum lipid profiles in overweight patients with hyperlipidemia: a double-blind randomized controlled trial. Sci Rep. 2015;5:10344. doi: 10.1038/srep10344.PubMedUsed to support: Human double-blind RCT (n=97, 150 mg/day mangiferin, 12 weeks) in overweight patients with diagnosed hyperlipidemia: significant reductions in triglycerides and free fatty acids, higher HDL cholesterol, and a lower insulin resistance index. The same trial found no difference versus placebo in total cholesterol, LDL cholesterol, blood glucose or insulin, so it does not support cholesterol, LDL or blood sugar claims. It tested generic mangiferin, not the Melostacio brand, in a disease population rather than healthy consumers.
  2. Jyotshna, Khare P, Shanker K Mangiferin: A review of sources and interventions for biological activities. Biofactors. 2016;42(5):504-514. doi: 10.1002/biof.1308.PubMedUsed to support: Narrative review of mangiferin sources and its reported antioxidant, anti-inflammatory and metabolic activities. A review is not new clinical evidence, and most of the underlying work is laboratory and animal research, so it supports background and proposed mechanisms only, not human benefit claims.
  3. Wu Y, Liu W, Yang T, Li M, Qin L, Wu L, Liu T Oral administration of mangiferin ameliorates diabetes in animal models: a meta-analysis and systematic review. Nutr Res. 2021;87:57-69. doi: 10.1016/j.nutres.2020.12.017.PubMedUsed to support: Systematic review and meta-analysis of 19 preclinical studies showing mangiferin significantly reduces blood glucose (SMD -1.27) and improves glycolipid metabolism via anti-inflammatory and antioxidative mechanisms. Note: animal model evidence; human RCT data are limited. Cited for mechanistic basis of glucose management benefit.