Phenylpiracetam (Phenotropil / Carphedon)

Synthetic compound: phenyl-substituted piracetam, developed in Russia
Evidence Level
Preliminary
3 Clinical Trials
6 Documented Benefits
1/5 Evidence Score

Phenylpiracetam (sold in Russia as Phenotropil) is a prescription medicine, not a dietary supplement. It is not an approved drug in the US, UK or EU, and it does not meet the legal definition of a dietary supplement ingredient in those markets. Chemically it is a synthetic, phenyl-substituted version of piracetam with stimulant-like effects. Carphedon, its sport-testing name, is on the World Anti-Doping Agency Prohibited List as a stimulant, so any tested athlete who takes it risks a doping violation. The only two studies cited on this page are small Russian-language trials in stroke patients undergoing rehabilitation. There is no controlled evidence in healthy people and no long-term safety data.

Studied Dose No dose has been established for healthy people. The two human studies cited here were done in hospital patients recovering from stroke, under medical supervision. Figures of roughly 100 to 200 mg a day that circulate online come from user communities, not from controlled trials.
Active Compound Phenylpiracetam ((R,S)-2-(2-oxo-4-phenyl-1-pyrrolidinyl)acetamide; fonturacetam, carphedon, phenotropil) — phenyl-substituted piracetam.

Benefits

Studied only in stroke patients, not in healthy people

The only human research cited on this page is two small Russian-language studies in people recovering from a stroke, published in 2005 and 2010 in a Russian neurology and psychiatry journal. They reported improvement in neurological deficits and in cognitive function in those patients. Stroke rehabilitation is specialist medical care, and results there say nothing about what this compound does for a healthy person. Neither study is available in full in English, so group sizes, randomization and blinding cannot be checked.

Fatigue and low energy: not supported by the studies cited here

No study cited on this page tests phenylpiracetam for everyday tiredness, chronic fatigue syndrome or fatigue after head injury. Both references are stroke rehabilitation trials. Russian regulators do list fatigue-type conditions among the approved uses of the prescription medicine Phenotropil, but a regulatory listing in one country is not evidence you can check, and none of it applies to a healthy person looking for more energy.

Origins in the Soviet space program

Phenylpiracetam was developed in the Soviet Union in the 1980s, and its reported use in the space program is part of its history rather than evidence of a benefit. No study cited on this page measured stamina, cold tolerance or mental performance in healthy people. Being banned in sport is an anti-doping classification decision, not proof that the compound improves performance.

Cognitive problems after stroke: a supervised medical use, not a consumer one

The evidence cited here covers one situation only: people recovering from a stroke, treated in a Russian medical setting. No study on this page involves head injury, brain surgery or any other cause of cognitive decline. Stroke and brain injury need specialist care, and nothing here is a reason for a healthy person to take this compound for memory or focus.

Epilepsy: no verifiable study is cited

The reference list on this page contains no epilepsy study. Any use alongside anti-seizure medication belongs to Russian prescribing practice under a neurologist's supervision. People with epilepsy should never add or change anything without their doctor, since stimulant-like compounds and seizure medicines can interact.

Banned in sport: doping violation risk

Carphedon, the sport-testing name for phenylpiracetam, is on the World Anti-Doping Agency Prohibited List as a stimulant, and athletes have been sanctioned for it. If you are drug tested at any level, taking this risks a doping violation. Appearing on a banned list is a regulatory classification, not evidence that it makes anyone faster or stronger.

Mechanism of action

1

Dopamine reuptake inhibition (stimulant mechanism)

Laboratory and rodent work suggests phenylpiracetam slows the reuptake of dopamine, which sets it apart from other racetams and may explain its stimulant-like feel. The finding on effort-based responding comes from rats. None of this has been shown to produce a measurable benefit in people, and a mechanism is not evidence of an effect.

2

Multi-receptor neurotransmitter modulation

Laboratory work suggests it also affects several other brain signalling systems, and the added phenyl group appears to help it cross into the brain more readily than piracetam. These are preclinical observations. They do not demonstrate calming, cognitive or brain-protective effects in people, and no human study on this page tested any of them.

3

Locomotor activity stimulation

In rodents, phenylpiracetam increases movement and activity in a way that resembles a mild stimulant, with one mirror-image form more active than the other. These are animal findings. More movement in a cage is not the same as better physical performance in a person.

4

Cold tolerance: claimed, not demonstrated here

Cold tolerance is often mentioned in accounts of this compound's origins, but no study cited on this page measured it, in animals or in people. Treat it as an unverified claim.

5

Brain protection: animal models only

Animal models of reduced blood flow to the brain have been used to compare phenylpiracetam with piracetam. Those are laboratory models in animals, not people. Russian doctors do prescribe it after stroke, but the two human studies cited here are small, Russian-language, and cannot be checked in detail from their English abstracts.

Clinical trials

1
Russian report in vascular brain disease (not in this page's verified reference list)

Russian-language report attributed to Gustov and colleagues, 2006, in Zh Nevrol Psikhiatr Im S S Korsakova. No PubMed ID is given for it, and it is not one of the two references listed on this page.

Hospital patients with blood-vessel-related brain disease, treated under medical care. The number of participants, how they were assigned to groups and whether anyone was blinded are not available in English.

The report describes reduced neurological deficits and better memory and attention compared with a control group. Because the full text is Russian-language and no PubMed ID is provided, the result cannot be independently checked, group sizes are unknown, and it was conducted in patients under medical care rather than in healthy adults.

2
Russian epilepsy report (not in this page's verified reference list)

Russian-language report attributed to Lybzikova and colleagues, 2008, in Zh Nevrol Psikhiatr Im S S Korsakova. No PubMed ID is given, and it is not among the two references listed on this page.

People with diagnosed epilepsy already taking anti-seizure medication, treated by doctors. The number of participants and the study design are not available in English.

The report describes fewer seizures and better cognitive function. It cannot be verified, no control group or blinding is described in what is available in English, and it concerns a diagnosed medical condition managed with prescription drugs. Nothing here applies to a healthy person.

3
Animal pharmacology: R and S forms compared in rodents

Preclinical pharmacology study (Zvejniece L, Svalbe B, Veinberg G, Grinberga S, Vorona M, Kalvinsh I, Basic Clin Pharmacol Toxicol 109(5):407-412, doi:10.1111/j.1742-7843.2011.00742.x).

Rodents, not people. The two mirror-image forms of phenylpiracetam were compared for movement, behaviour in a depression-type test, and memory tasks.

In rats, the R form increased movement at 10 to 50 mg/kg and produced antidepressant-type effects in a behavioural test at 50 to 100 mg/kg, and it was more active than the S form. These are animal doses and animal behaviour tests. They do not show that phenylpiracetam lifts mood or boosts energy in people, and no human mood study is cited on this page.

Side effects and drug interactions

Common Potential side effects

Not a dietary supplement: this is a prescription medicine in Russia and is neither an approved drug nor a legal supplement ingredient in the US, UK or EU. Stimulant-type effects reported include insomnia, agitation, irritability, anxiety, restlessness and headache.
Users commonly report that the effects fade within one to two weeks of daily use. This comes from user reports, not from trial data.
GI upset (nausea).
Can raise blood pressure and heart rate, as stimulant-like compounds do. Anyone with heart problems or high blood pressure should avoid it.
Athletes: WADA-PROHIBITED — will fail drug tests in competition (Section S6 Stimulants).
Pregnancy/lactation: avoid.
Anxiety disorders, bipolar disorder or psychosis: avoid. It is stimulating and may worsen symptoms. Do not combine it with psychiatric medication without medical supervision.
No established long-term safety data in healthy people. The two human studies cited here were short, done in stroke patients, and carried out under medical supervision.

Important Drug interactions

MAOIs: significant interaction risk (dopaminergic effects).
Stimulants such as caffeine and ADHD medication: effects can add up, raising the risk of insomnia, agitation, high blood pressure and a fast heart rate.
Antidepressants: interactions are possible and have not been studied. Do not combine without medical supervision.
Sympathomimetic decongestants: additive cardiovascular effects.
Anti-seizure medication: unpredictable. It is used alongside these drugs in Russia under specialist supervision, but a stimulant-like compound should never be added to a seizure treatment plan on your own.
Do not assume it is safe alongside other medicines. Interaction data in healthy people is essentially absent, and where it is legal at all it is a prescription-only medicine. Check with a doctor or pharmacist before combining it with anything.

Frequently asked questions about Phenylpiracetam (Phenotropil / Carphedon)

What is phenylpiracetam?

Phenylpiracetam, also called Phenotropil or carphedon, is a synthetic compound related to piracetam, with an added phenyl group that makes it more stimulating. It is a prescription medicine in Russia and is not an approved drug or a legal dietary supplement ingredient in the US, UK or EU. It is also banned in sport by the World Anti-Doping Agency. The only human studies cited on this page are Russian trials in stroke patients.

Why is phenylpiracetam banned in sports?

The World Anti-Doping Agency lists carphedon (phenylpiracetam) as a prohibited stimulant. Any athlete subject to testing who takes it risks a doping violation, whether or not it actually does anything for performance.

How much phenylpiracetam is used?

There is no established dose for healthy people. Figures of around 100 to 200 mg a day come from user communities, not from controlled trials. Product quality varies widely, and in most Western countries it is not a legal supplement ingredient at all.

Is phenylpiracetam safe?

Its safety in healthy people has not been established. Reported effects include overstimulation, agitation, irritability, trouble sleeping, and raised blood pressure and heart rate, and there is no long-term safety data. It is a prescription medicine in Russia, is not an approved drug or a legal supplement ingredient in the US, UK or EU, and is banned in sport. Anyone considering it should speak with a healthcare professional first.

What is Phenylpiracetam used for?

Phenylpiracetam is researched primarily for Cognitive. The only human research cited on this page is two small Russian-language studies in people recovering from a stroke, published in 2005 and 2010 in a Russian neurology and psychiatry journal.

What is the recommended dosage of Phenylpiracetam?

The clinically studied dose is No dose has been established for healthy people. The two human studies cited here were done in hospital patients recovering from stroke, under medical supervision. Always follow the product label and check with a healthcare provider for personal advice.

Is Phenylpiracetam safe, and does it have side effects?

For most healthy adults, Phenylpiracetam is well tolerated at studied doses. Reported effects can include: Not a dietary supplement: this is a prescription medicine in Russia and is neither an approved drug nor a legal supplement ingredient in the US, UK or EU. Stimulant-type effects reported include insomnia, agitation, irritability, anxiety, restlessness and headache. It may also interact with some medications. Phenylpiracetam is not right for everyone, so check with a healthcare provider first if you are pregnant or breastfeeding, have a medical condition, or take prescription medication.

Does Phenylpiracetam interact with any medications?

Possible interactions include: MAOIs: significant interaction risk (dopaminergic effects). Stimulants such as caffeine and ADHD medication: effects can add up, raising the risk of insomnia, agitation, high blood pressure and a fast heart rate. If you take prescription medication, check with a pharmacist or doctor before using it.

How strong is the scientific evidence for Phenylpiracetam?

NutraSmarts rates the evidence for Phenylpiracetam as Preliminary (1 out of 5). It is backed by 3 clinical trials and 2 cited references summarized on this page. A higher rating reflects more, larger, and better-designed human studies.

References(2 citations)

Evidence ratings on NutraSmarts are based on the totality of human clinical research, with emphasis on randomized controlled trials, meta-analyses, and systematic reviews. The references below directly support claims made throughout this page.

  1. Koval'chuk VV, Skoromets AA, Koval'chuk IV, Stoianova EG, Vysotskaia ML, Melikhova EV, Il'iaĭnen EV [Efficacy of phenotropil in the rehabilitation of stroke patients] Zh Nevrol Psikhiatr Im S S Korsakova. 2010;110(12 Pt 2):38-40.PubMedUsed to support: Russian-language clinical study indexed in PubMed, evaluating phenotropil during stroke rehabilitation and reporting improvement in neurological deficits and cognitive function in those patients. It supports supervised use in stroke rehabilitation only. It does not support any benefit for cognition, energy, mood or stress in healthy people.
  2. Gerasimova MM, Chichanovskaia LV, Slezkina LA [The clinical and immunological aspects of the effects of phenotropil on consequences of stroke] Zh Nevrol Psikhiatr Im S S Korsakova. 2005;105(5):63-4.PubMedUsed to support: Russian-language clinical study in patients with after-effects of stroke, reporting clinical and immune-system outcomes. This is medical treatment of stroke survivors and is not evidence of a benefit for a healthy consumer. It is one of only two human studies cited on this page.