Leucoselect® Phytosome (Grape Seed Phytosome — Indena)

Vitis vinifera
Evidence Level
Limited
2 Clinical Trials
5 Documented Benefits
2/5 Evidence Score

Leucoselect® Phytosome is a grape seed extract phytosome® developed by Indena (Italy) — using Phytosome® technology applied to grape seed proanthocyanidins (OPCs). It is sold for antioxidant and cardiovascular support, but the published human work on this branded extract is small: a 1998 study of a blood antioxidant marker, a 2003 randomized crossover study of how easily LDL cholesterol oxidized in heavy smokers, and a 2014 observational report in frail elderly people. No cited study compared its absorption head to head against standard grape seed extract, and none measured blood pressure, endothelial function, cholesterol levels, or heart events.

Studied Dose 100-300 mg/day, the range used in the small human studies available
Active Compound Grape seed oligomeric proanthocyanidins (OPCs) Phytosome® formulation

Benefits

Cardiovascular and Vascular Function

In a small randomized crossover study in heavy smokers, a standardized grape seed extract reduced how easily LDL cholesterol was oxidized in a laboratory test. That is a marker of oxidative stress, not a measure of heart health, and it was studied in a high risk group. None of the cited studies measured endothelial function, blood pressure, or cardiovascular events.

Antioxidant Activity

Grape seed proanthocyanidins act as antioxidants. In a small 1998 study, co authored by staff of the manufacturer, Leucoselect raised a serum antioxidant marker in volunteers. That is a blood measurement, not a demonstrated health outcome.

Microcirculation Support

None of the cited studies measured microcirculation or capillary permeability in people, so this remains a proposed effect rather than a demonstrated one.

What the LDL Oxidation Study Actually Measured

The 2003 study looked at how resistant LDL cholesterol was to oxidation in heavy smokers, not at whether cholesterol levels themselves improved. No cited trial reported changes in total cholesterol, LDL, HDL, or triglycerides.

Phytosome Delivery Format (Not a Health Benefit)

Phytosome is a format that pairs plant compounds with phospholipids, and the maker says this improves absorption. No head to head absorption study comparing Leucoselect Phytosome with standard grape seed extract is cited here, so treat that comparison as a manufacturer claim rather than a settled finding. A delivery format is also not a health benefit on its own.

Mechanism of action

1

OPC Antioxidant Activity

Grape seed proanthocyanidins can neutralize free radicals in laboratory testing and may help recycle vitamins C and E. This is standard antioxidant chemistry, not proof of a specific health effect in people.

2

Phytosome® Bioavailability Enhancement

Proanthocyanidins are poorly and variably absorbed. The phytosome format is intended to improve absorption, though no head to head absorption comparison is cited on this page.

3

Endothelial Nitric Oxide Support

Proposed only: grape seed compounds may support nitric oxide production in the lining of blood vessels. None of the studies cited here measured nitric oxide or endothelial function.

4

Capillary Integrity

Proanthocyanidins are proposed to reduce leakiness of small blood vessels. This was not measured in the human studies cited here, and this ingredient is not offered as a treatment for vein conditions.

Clinical trials

1
LDL Oxidation Marker in Heavy Smokers (2003)

A small randomized crossover study of a standardized grape seed extract, published in Metabolism in 2003. Several authors were affiliated with the manufacturer, Indena.

Heavy smokers, chosen because smoking raises oxidative stress. Small sample.

LDL cholesterol became more resistant to oxidation in a laboratory test. That is a surrogate marker. Vascular function, blood pressure, and cholesterol levels were not shown to improve.

2
Other Published Leucoselect Research

No pooled analysis of Leucoselect Phytosome is cited. The remaining published work is a 1998 study of a serum antioxidant marker, a 2014 descriptive observational report with no randomization and no control group, and a 2016 laboratory paper.

Small groups of healthy volunteers and frail elderly people with inflammatory and allergic conditions, plus human cells studied in a laboratory.

The 1998 study reported a change in a blood antioxidant marker. The 2014 report described immune measurements but, without a control group, cannot show cause and effect. The 2016 paper tested grape seed procyanidin extract on human lung cancer cell lines and airway cells in the laboratory; that is early bench research, not evidence that this supplement prevents or treats cancer.

Side effects and drug interactions

Common Potential side effects

Generally well-tolerated.
Mild GI distress.
Allergic reactions to grape rare.
Theoretical bleeding at high doses.
Soy allergy considerations (Phytosome).

Important Drug interactions

Anticoagulants — modest antiplatelet effects.
Antihypertensives — modest BP effects.
Pregnancy and breastfeeding: there is not enough data on concentrated grape seed extract, so ask your doctor before using it.
Pre-surgery — discontinue 1-2 weeks.
Soy allergy — Phytosome consideration.

Frequently asked questions about Leucoselect® Phytosome (Grape Seed Phytosome — Indena)

What is Leucoselect Phytosome?

Leucoselect® Phytosome is a grape seed extract phytosome® developed by Indena (Italy) — using Phytosome® technology applied to grape seed proanthocyanidins (OPCs).

What is Leucoselect Phytosome used for?

Leucoselect Phytosome is researched primarily for Cardiovascular and Antioxidant. In a small randomized crossover study in heavy smokers, a standardized grape seed extract reduced how easily LDL cholesterol was oxidized in a laboratory test.

What is the recommended dosage of Leucoselect Phytosome?

The clinically studied dose is 100-300 mg/day, the range used in the small human studies available Always follow the product label and check with a healthcare provider for personal advice.

Is Leucoselect Phytosome safe, and does it have side effects?

For most healthy adults, Leucoselect Phytosome is well tolerated at studied doses. Reported effects can include: Generally well-tolerated. Mild GI distress. It may also interact with some medications. Leucoselect Phytosome is not right for everyone, so check with a healthcare provider first if you are pregnant or breastfeeding, have a medical condition, or take prescription medication.

Does Leucoselect Phytosome interact with any medications?

Possible interactions include: Anticoagulants — modest antiplatelet effects. Antihypertensives — modest BP effects. If you take prescription medication, check with a pharmacist or doctor before using it.

How strong is the scientific evidence for Leucoselect Phytosome?

NutraSmarts rates the evidence for Leucoselect Phytosome as Limited (2 out of 5). It is backed by 2 clinical trials and 4 cited references summarized on this page. A higher rating reflects more, larger, and better-designed human studies.

References(4 citations)

Evidence ratings on NutraSmarts are based on the totality of human clinical research, with emphasis on randomized controlled trials, meta-analyses, and systematic reviews. The references below directly support claims made throughout this page.

  1. Nuttall SL, Kendall MJ, Bombardelli E, Morazzoni P An evaluation of the antioxidant activity of a standardized grape seed extract, Leucoselect J Clin Pharm Ther. 1998;23(5):385-389. doi: 10.1046/j.1365-2710.1998.00180.x.PubMedUsed to support: Measured a serum antioxidant marker in humans, which is a blood biomarker rather than a clinical outcome. Small, early, and co authored by staff of the manufacturer Indena (Bombardelli, Morazzoni). Preliminary.
  2. Vigna GB, Costantini F, Aldini G, Carini M, Catapano A, Schena F, Tangerini A, Zanca R, Bombardelli E, Morazzoni P, Mezzetti A, Fellin R, Maffei Facino R Effect of a standardized grape seed extract on low-density lipoprotein susceptibility to oxidation in heavy smokers Metabolism. 2003;52(10):1250-1257. doi: 10.1016/s0026-0495(03)00192-6.PubMedUsed to support: Randomized crossover study showing that LDL cholesterol became less easily oxidized in heavy smokers. That is a surrogate laboratory marker, not a cardiovascular outcome, and the study was small with authors affiliated with Indena.
  3. Magrone T, Pugliese V, Fontana S, Jirillo E Human use of Leucoselect Phytosome with special reference to inflammatory-allergic pathologies in frail elderly patients Curr Pharm Des. 2014;20(6):1011-1019. doi: 10.2174/138161282006140220144411.PubMedUsed to support: A descriptive observational report on Leucoselect Phytosome use in frail elderly patients with inflammatory and allergic conditions. It was not randomized and had no control group, so it cannot show that the supplement caused any change.
  4. Mao JT, Smoake J, Park HK, Lu QY, Xue B Grape Seed Procyanidin Extract Mediates Antineoplastic Effects against Lung Cancer via Modulations of Prostacyclin and 15-HETE Eicosanoid Pathways Cancer Prev Res (Phila). 2016;9(12):925-932. doi: 10.1158/1940-6207.CAPR-16-0122.PubMedUsed to support: Laboratory research using human premalignant and malignant lung cell lines plus cells collected from airway lavage. This is early bench work on possible anti-inflammatory pathways, not a clinical trial, and it does not show that the supplement prevents or treats lung cancer in people.