Lactoperoxidase (LPO Salivary Enzyme System)

Lactoperoxidase (LPO) — bovine + human salivary enzyme
Evidence Level
Limited
3 Clinical Trials
7 Documented Benefits
2/5 Evidence Score

A salivary peroxidase enzyme: a heme glycopeptide of approximate mass ~78,000 Da (bovine) / ~80,000 Da (human) with a calcium-binding site (Asp227) and an autocatalytic heme B center. It oxidizes salivary thiocyanate (SCN-) in the presence of H2O2 to hypothiocyanite, a broad-spectrum antimicrobial. All human evidence is oral-care that acts locally in the mouth: toothpaste (rinse-and-spit) and oral tablets that dissolve in the mouth. Trials of an LPO toothpaste three-enzyme system (amyloglucosidase + glucose oxidase + LPO) with lactoferrin and lysozyme, and of lactoferrin + LPO oral tablets, reduced gingival inflammation and plaque, and a systematic review of three small studies reached the same conclusion. There is no evidence for LPO as a swallowed systemic supplement, and none for hair, skin, or nail outcomes. Bovine LPO is structurally and functionally similar to human salivary LPO.

Studied Dose Oral lozenge tablets: lactoferrin 60 mg + LPO 7.8 mg/day (or 20 mg + 2.6 mg). Most evidence is topical toothpaste (rinse-and-spit), not a swallowed dose.
Active Compound Lactoperoxidase (LPO); bovine and human salivary enzyme. Single-chain monomeric glycopeptide ~78-80 kDa with autocatalytic heme B and Ca2+-binding site (Asp227).

Benefits

Gingival index reduction LF + LPO tablets

In a randomized double-blind placebo-controlled trial in healthy adults, high-dose tablets (lactoferrin 60 mg/d + LPO 7.8 mg/d) significantly reduced the Gingival Index vs placebo. These oral tablets dissolve in and act locally in the mouth, and the single trial was funded by the tablet maker (Morinaga Milk Industry), with efficacy analyzed in 109 of 150 randomized adults.

Toothpaste enzyme system gingivitis 13-week RCT

A double-blind randomized parallel-group home-use RCT in healthy non-smokers tested a toothpaste containing enzymes (amyloglucosidase + glucose oxidase + LPO) plus proteins (lactoferrin + lysozyme), reflecting natural saliva composition, vs a commercial control. The three-enzyme system reproduces the natural salivary defense mechanism rather than introducing exogenous antimicrobials.

Plaque and gingivitis in xerostomia

In patients with radiation-induced xerostomia, LPO toothpaste reduced the rate of supragingival plaque formation, and gingival inflammation was lower. Particularly relevant population, since xerostomia patients have impaired natural salivary defense. This was a single-blind pilot crossover in only 12 patients using an LPO toothpaste (topical, rinse-and-spit), which limits any firm conclusion.

Hypothiocyanite antimicrobial production (mechanism)

LPO oxidizes salivary thiocyanate (SCN⁻) using H₂O₂ as cofactor to generate hypothiocyanite (OSCN⁻) — a broad-spectrum antimicrobial active against both Gram-positive and Gram-negative pathogens. This defense pathway is delivered locally by LPO oral-care products (toothpaste and dissolving tablets), not by systemic supplementation.

Three-enzyme synergistic system

Amyloglucosidase + glucose oxidase generate H₂O₂ from glucose, which LPO then uses with thiocyanate to produce hypothiocyanite. Self-sustaining enzyme cascade — provides continuous low-level antimicrobial activity from dietary glucose substrate without exogenous H₂O₂ delivery.

Oral microbiome rebalancing (proposed mechanism)

Hypothiocyanite exerts selective antimicrobial pressure that could favor commensal species over periodontal pathogens rather than acting as a blanket antibacterial. This is a proposed mechanism: the cited oral-care trials measured gingival and plaque scores, not oral-microbiome composition, and none reports a Neisseria increase.

Systematic review (D'Agostino & Dolci, 2025)

A systematic review found that toothpaste with amyloglucosidase + glucose oxidase + LPO + lysozyme + lactoferrin is effective for preventing gingivitis and managing gingival inflammation short-term and long-term, via reduced MGI, BI, and PI scores. Honest limitation acknowledged in the review: limited number of eligible studies.

Mechanism of action

1

Hypothiocyanite generation (LPO-SCN-H₂O₂ system)

The core LPO mechanism: oxidation of thiocyanate using H₂O₂ as cofactor to generate hypothiocyanite, a broad-spectrum antimicrobial. The natural salivary defense pathway.

2

Three-enzyme synergistic system

Amyloglucosidase + glucose oxidase cascade generates H₂O₂ from dietary glucose, which LPO uses to produce hypothiocyanite. Self-sustaining cascade providing continuous low-level antimicrobial activity.

3

Gram-positive and Gram-negative pathogen inhibition

Hypothiocyanite has broad-spectrum activity against periodontal pathogens including Streptococcus mutans, Porphyromonas gingivalis, and Aggregatibacter actinomycetemcomitans — covering the major Gram-positive and Gram-negative oral pathogens.

4

Heme B catalytic center + calcium binding

LPO contains an autocatalytic heme B center for the peroxidation reaction plus a calcium-binding site (Asp227) supporting structural stability. Standard heme peroxidase pharmacology with LPO-specific substrate preferences.

5

Oral microbiome shift toward health

In the mouth, selective pressure appears to favor commensal species (e.g., Neisseria) over periodontal pathogens, rebalancing the ORAL microbiome rather than acting as a blanket antibacterial. This is a local oral-cavity effect.

6

Salivary defense system reproduction

The natural salivary LPO plus thiocyanate plus H₂O₂ system can be reinforced LOCALLY by LPO-containing oral-care products (toothpaste, lozenges), which may help in xerostomia where saliva is reduced. This is a local oral-cavity effect, not systemic supplementation.

Clinical trials

1
Oral LF + LPO Tablets (dissolve and act locally in the mouth), 12-Week RCT
PubMed

Clinical evidence on Lactoperoxidase (LPO Salivary Enzyme System) for the indications and outcomes described.

healthy adults

Nakano M et al. 2019 (authors employed by Morinaga Milk Industry, which makes the tablets). Randomized double-blind placebo-controlled trial: 150 adults randomized, 109 analyzed for efficacy. High-dose tablets (lactoferrin 60 mg/d + LPO 7.8 mg/d) for 12 weeks significantly reduced the Gingival Index vs placebo. These are oral tablets that act locally in the mouth on gum inflammation, not a systemically absorbed supplement.

2
Enzyme/Protein Toothpaste Gingivitis 13-Week Clinical Trial
PubMed

13-week double-blind randomized parallel-group home-use clinical trial in healthy non-smokers (mean MGI 2.00-2.75).

Clinical population described in trial publication.

13-week double-blind randomized parallel-group home-use clinical trial in healthy non-smokers (mean MGI 2.00-2.75). Toothpaste with a three-enzyme system (amyloglucosidase + glucose oxidase + LPO) plus lactoferrin and lysozyme vs commercial control (229 completed; study co-authored and funded by Unilever Oral Care). This is a rinse-and-spit toothpaste applied topically to the oral cavity, not a swallowed supplement.

3
LPO Toothpaste (topical, rinse-and-spit) Xerostomia 52-Day Pilot Crossover, n=12
PubMed

Single-blind crossover 52-day trial in 12 patients with radiation-induced xerostomia.

12 patients with radiation-induced xerostomia

Single-blind crossover 52-day trial in 12 patients with radiation-induced xerostomia. LPO toothpaste reduced rate of supragingival plaque formation; gingival inflammation was lower. Small sample size in a clinically important population (xerostomia patients).

Side effects and drug interactions

Common Potential side effects

Generally well-tolerated; topical/oral application of natural enzyme system.
Mild oral irritation (rare, transient).
Allergic reactions (rare; bovine-derived).
Pregnancy/lactation: limited specific data; toothpaste application generally considered safe.
Long-term safety: multiple multi-week toothpaste/tablet trials supportive.
Dry mouth (xerostomia): well-tolerated + beneficial population per PMID 8063434.
Bovine-derived ingredient sensitivities: caution.

Important Drug interactions

Topical/oral application — minimal systemic absorption.
Most medications: no documented interactions.
Fluoride toothpaste: compatible — typically formulated together.
Antibiotics (topical or systemic): theoretical complementary antimicrobial activity.
Mouthwash/oral antiseptics: avoid concurrent use within 30 minutes (potential enzyme inactivation).

Frequently asked questions about Lactoperoxidase (LPO Salivary Enzyme System)

What is lactoperoxidase?

Lactoperoxidase is a natural enzyme found in milk, saliva, and other secretions that has antibacterial activity. It is part of the body's innate defense and is used in some oral-care products and as a natural preservative.

What is lactoperoxidase used for?

It is used mainly in oral-care products (toothpastes and mouthwashes for dry mouth) and as a natural antimicrobial preservative in foods; its studied effects are local to the mouth, not systemic.

How is lactoperoxidase taken?

It is most often delivered through oral-care products or specific formulas rather than as a standalone supplement; follow the specific product's directions.

Is lactoperoxidase safe?

It is a natural enzyme found in milk and saliva and is generally regarded as safe. Because it is typically dairy-derived, those with milk allergies should check product sourcing.

What is the recommended dosage of Lactoperoxidase?

The clinically studied dose is Oral lozenge tablets: lactoferrin 60 mg + LPO 7.8 mg/day (or 20 mg + 2.6 mg). Most evidence is topical toothpaste (rinse-and-spit), not a swallowed dose. Always follow the product label and check with a healthcare provider for personal advice.

Is Lactoperoxidase safe, and does it have side effects?

For most healthy adults, Lactoperoxidase is well tolerated at studied doses. Reported effects can include: Generally well-tolerated; topical/oral application of natural enzyme system. Mild oral irritation (rare, transient). It may also interact with some medications. Lactoperoxidase is not right for everyone, so check with a healthcare provider first if you are pregnant or breastfeeding, have a medical condition, or take prescription medication.

Does Lactoperoxidase interact with any medications?

Possible interactions include: Topical/oral application — minimal systemic absorption. Most medications: no documented interactions. If you take prescription medication, check with a pharmacist or doctor before using it.

How strong is the scientific evidence for Lactoperoxidase?

NutraSmarts rates the evidence for Lactoperoxidase as Limited (2 out of 5). It is backed by 3 clinical trials and 6 cited references summarized on this page. A higher rating reflects more, larger, and better-designed human studies.

References(6 citations)

Evidence ratings on NutraSmarts are based on the totality of human clinical research, with emphasis on randomized controlled trials, meta-analyses, and systematic reviews. The references below directly support claims made throughout this page.

  1. Nakano M, Yoshida A, Wakabayashi H, Tanaka M, Yamauchi K, Abe F, Masuda Y Effect of tablets containing lactoferrin and lactoperoxidase on gingival health in adults: A randomized, double-blind, placebo-controlled clinical trial J Periodontal Res. 2019;54(6):702-708. doi: 10.1111/jre.12679.PubMedUsed to support: Randomized double-blind placebo-controlled trial (150 adults randomized, 109 analyzed for efficacy) of oral tablets containing lactoperoxidase 7.8 mg/day plus lactoferrin 60 mg/day for 12 weeks. The high-dose group had a significant reduction in the Gingival Index versus placebo. The tablets act locally in the mouth on gum inflammation; the trial did not measure any digestive or systemic immune outcome, and the authors were employed by the tablet maker (Morinaga Milk Industry).
  2. Hu X, Zhang P, Zhang L, Matheson JR, Lin S, Sun JN, Delfanti C, Tian J, Gupta AK, Vasantharaghavan R, Huang R The effect of enzyme and protein containing toothpaste on gingival condition: a randomised controlled study BMC Oral Health. 2025;25(1):1727. doi: 10.1186/s12903-025-07096-7.PubMedUsed to support: 26-week double-blind randomized controlled trial in a Chinese adult population of a rinse-and-spit fluoride toothpaste containing lysozyme, lactoperoxidase, and lactoferrin versus a control fluoride toothpaste. The test toothpaste significantly improved gingival index and reduced supragingival plaque. This is a topical oral-care product, and the study was co-authored and funded by Unilever Oral Care.
  3. van Steenberghe D, Van den Eynde E, Jacobs R, Quirynen M Effect of a lactoperoxidase containing toothpaste in radiation-induced xerostomia Int Dent J. 1994;44(2):133-138.PubMedUsed to support: Controlled human clinical study (n=12) of LPO-containing toothpaste in patients with radiation-induced xerostomia (dry mouth), assessing plaque, gingival inflammation, and subgingival microbiota — supporting plaque and gingivitis in xerostomia claim.
  4. Tenovuo J Clinical applications of antimicrobial host proteins lactoperoxidase, lysozyme and lactoferrin in xerostomia: efficacy and safety Oral Dis. 2002;8(1):23-29. doi: 10.1034/j.1601-0825.2002.1o781.x.PubMedUsed to support: Clinical review evaluating LPO, lysozyme, and lactoferrin incorporated into oral care products (dentifrices, mouthrinses, gels) to restore salivary antimicrobial capacity in xerostomia — supporting three-enzyme synergistic system, hypothiocyanite antimicrobial production mechanism, and clinical applications for plaque/gingivitis in dry mouth.
  5. Daly S, Seong J, Newcombe R, Davies M, Nicholson J, Edwards M, West N A randomised clinical trial to determine the effect of a toothpaste containing enzymes and proteins on gum health over 3 months J Dent. 2019;80 Suppl 1:S26-S32.PubMedUsed to support: 13-week (3-month) double-blind randomized parallel-group home-use RCT in healthy non-smokers (mean MGI 2.00-2.75) of a toothpaste with the three-enzyme system (amyloglucosidase + glucose oxidase + lactoperoxidase) plus lactoferrin and lysozyme vs commercial control, showing significantly better gingival and plaque scores — the pivotal described trial for the toothpaste enzyme-system gingivitis 13-week benefit and the three-enzyme synergistic system.
  6. D'Agostino S, Dolci M Exploring the Effect of Enzyme and Protein-Containing Toothpaste on Gum Health: A Systematic Review Microorganisms. 2025;13(5):1158.PubMedUsed to support: Systematic review concluding that toothpaste containing amyloglucosidase + glucose oxidase + lactoperoxidase + lysozyme + lactoferrin is effective for preventing gingivitis and managing gingival inflammation short- and long-term (reduced MGI, BI, PI), with the honest limitation of few eligible studies — the systematic review referenced in the summary at the top of this page and the systematic-review benefit.