Bergavit® (Bergamot Flavonoid Extract — Bionap)

Citrus bergamia
Evidence Level
Limited
1 Clinical Trial
3 Documented Benefits
2/5 Evidence Score

Bergavit® is a standardized bergamot (Citrus bergamia) fruit extract from Bionap, made by concentrating the flavonoids from bergamot juice, with neohesperidin, naringin and neoeriocitrin as its markers at about 47, 37 and 16 percent of the flavonoid content in the studied material. Bergamot also contains brutieridin and melitidin, two flavonoids with a statin-like fragment, but they are not what the extract is standardized to. Bergamot flavonoids are studied for supporting healthy cholesterol and triglyceride levels. The study of this branded extract described on this page followed 80 people for 6 months with no placebo group, so its numbers show change over time rather than an effect measured against a comparison group.

Studied Dose About 150 mg of bergamot flavonoids per day, the amount given for 6 months in the study described on this page.
Active Compound Bergamot fruit flavonoid extract standardized to its three main juice flavonoids, neohesperidin, naringin and neoeriocitrin (brutieridin and melitidin occur in bergamot but are not part of the standardization).

Benefits

Healthy cholesterol levels

In a 6 month study of 80 adults with higher than ideal cholesterol, everyone took the extract and there was no placebo group. Average total cholesterol fell from about 255 to 224 mg/dl, LDL from about 178 to 143 mg/dl and triglycerides from about 159 to 133 mg/dl, while HDL rose from about 50 to 54 mg/dl. Those are before and after figures within one group rather than a comparison against placebo.

Small dense LDL

In that same single group study, the LDL profile shifted away from the small, dense bands linked with cardiovascular risk. The largest of those bands, LDL-3, went from about 14.5 to 9.0 percent of total LDL, while the large LDL-1 band rose from about 41.2 to 49.6 percent. These are proportions of the LDL profile before and after, in a group with no placebo comparison.

Cardiovascular support

The same study measured carotid artery wall thickness by ultrasound and reported a drop from 1.2 to 0.9 mm over 6 months. That number deserves caution. Controlled trials of prescription cholesterol medicines typically shift carotid wall thickness by hundredths of a millimeter or less over a year, so a change of this size in half a year is far more than a study without a control group can support.

Mechanism of action

1

HMG-CoA reductase modulation

Brutieridin and melitidin carry a fragment resembling the active part of a statin, and laboratory work suggests they can inhibit HMG-CoA reductase, the enzyme that controls cholesterol synthesis. This is a proposed explanation from chemistry and cell studies rather than something measured in people, and these two flavonoids are not part of what the extract is standardized to.

2

Antioxidant flavonoids

The flavonoid mix is thought to limit oxidative modification of LDL and to support the lining of blood vessels. Neither was measured in the 6 month study cited on this page, so treat this as a proposed mechanism rather than a demonstrated one.

Clinical trials

1
Bergavit and Plasma Lipids: a 6 Month Single Group Study
PubMed

Six month prospective study of Bergavit at a fixed 150 mg of flavonoids daily, measuring plasma lipids, LDL subfractions and carotid artery wall thickness. Every participant received the extract. There was no placebo group and no randomization, and the authors list the missing control group as a limitation of their own work. (Toth et al., Frontiers in Pharmacology)

80 adults, mean age 55, with moderate hypercholesterolemia (LDL 160 to 190 mg/dl). 6 months, single group, no placebo.

Over 6 months, average total cholesterol fell from 6.6 to 5.8 mmol/l (about 255 to 224 mg/dl), LDL from 4.6 to 3.7 mmol/l (about 178 to 143 mg/dl) and triglycerides from 1.8 to 1.5 mmol/l (about 159 to 133 mg/dl), while HDL rose from 1.3 to 1.4 mmol/l (about 50 to 54 mg/dl). The share of LDL in the small, dense bands fell and large LDL rose. Carotid wall thickness was reported to fall from 1.2 to 0.9 mm. Every one of these is a before and after value inside a single group that all received the extract, so ordinary variation over time, seasonal change and any diet or lifestyle change the participants made are not separated out. The carotid figure in particular is far larger than what controlled trials of prescription cholesterol medicines produce in a year.

Side effects and drug interactions

Common Potential side effects

Generally well tolerated. The 6 month study reported no adverse events among its 80 participants, though that is a small and short safety record with no comparison group.
Mild heartburn or muscle cramps are occasionally reported by users of bergamot supplements rather than in the study cited here.
Citrus-sensitive individuals should start at a low dose.

Important Drug interactions

Statins: possible additive cholesterol lowering, so monitor with your doctor. This extract is not a replacement for a prescribed cholesterol medicine and is not a treatment for a lipid disorder, so do not stop or change a prescription on your own.
Drugs metabolized by CYP enzymes: bergamot, like grapefruit, contains compounds that can block CYP3A4 in the gut and raise blood levels of some medicines. How much of that carries over into a purified flavonoid extract is not established, so ask a pharmacist if any of your medicines carry a grapefruit warning.
Diabetes medication: blood sugar was not among the measurements in the study of this extract, but other bergamot preparations have been reported to affect it, so monitor.

Frequently asked questions about Bergavit® (Bergamot Flavonoid Extract — Bionap)

What is Bergavit?

Bergavit® is a standardized bergamot (Citrus bergamia) fruit extract from Bionap, made by concentrating the flavonoids from bergamot juice, with neohesperidin, naringin and neoeriocitrin as its markers at about 47, 37 and 16 percent of the flavonoid content in the studied material.

What is Bergavit used for?

Bergavit is researched primarily for Cardiovascular and Metabolic Health. In a 6 month study of 80 adults with higher than ideal cholesterol, everyone took the extract and there was no placebo group.

What is the recommended dosage of Bergavit?

The clinically studied dose is About 150 mg of bergamot flavonoids per day, the amount given for 6 months in the study described on this page. Always follow the product label and check with a healthcare provider for personal advice.

Is Bergavit safe, and does it have side effects?

For most healthy adults, Bergavit is well tolerated at studied doses. Reported effects can include: Generally well tolerated. The 6 month study reported no adverse events among its 80 participants, though that is a small and short safety record with no comparison group. It may also interact with some medications. Bergavit is not right for everyone, so check with a healthcare provider first if you are pregnant or breastfeeding, have a medical condition, or take prescription medication.

Does Bergavit interact with any medications?

Possible interactions include: Statins: possible additive cholesterol lowering, so monitor with your doctor. This extract is not a replacement for a prescribed cholesterol medicine and is not a treatment for a lipid disorder, so do not stop or change a prescription on your own. If you take prescription medication, check with a pharmacist or doctor before using it.

How strong is the scientific evidence for Bergavit?

NutraSmarts rates the evidence for Bergavit as Limited (2 out of 5). It is backed by 1 clinical trial and 2 cited references summarized on this page. A higher rating reflects more, larger, and better-designed human studies.

References(2 citations)

Evidence ratings on NutraSmarts are based on the totality of human clinical research, with emphasis on randomized controlled trials, meta-analyses, and systematic reviews. The references below directly support claims made throughout this page.

  1. Toth PP, Patti AM, Nikolic D, et al. Bergamot Reduces Plasma Lipids, Atherogenic Small Dense LDL, and Subclinical Atherosclerosis in Subjects with Moderate Hypercholesterolemia. Front Pharmacol. 2015;6:299..PubMedUsed to support: Six month single group study of Bergavit at 150 mg of flavonoids daily in 80 adults with moderate hypercholesterolemia. No placebo group and no randomization, so every result is a before and after comparison within one group.
  2. Spina A, Amone F, Zaccaria V, et al. Citrus bergamia Extract, a Natural Approach for Cholesterol and Lipid Metabolism Management: A Randomized, Double-Blind Placebo-Controlled Clinical Trial. Foods. 2024;13(23):3883..PubMedUsed to support: Randomized double-blind placebo-controlled trial of this branded extract at 150 mg of flavonoids daily for 4 months in 64 adults, reporting total cholesterol down 8.8 percent and LDL cholesterol down 11.5 percent against placebo. This is the controlled evidence the older single-group study lacked, and one author is an employee of the ingredient manufacturer.