Alpha-Ketoglutarate (AKG / Calcium AKG)

Endogenous TCA cycle intermediate
Evidence Level
Limited
3 Clinical Trials
6 Documented Benefits
2/5 Evidence Score

Alpha-ketoglutarate (AKG) is a compound central to the body's energy-producing Krebs cycle and to amino acid metabolism. It is used by athletes for performance and recovery, sometimes as arginine-AKG for blood-flow support, though the human trials are mixed: single-dose trials in trained and untrained men found no gain in strength, muscular endurance or blood flow, while one 8-week training study found a gain in bench press one-repetition maximum and peak anaerobic power. A calcium form (Ca-AKG) has drawn interest in longevity research, where it has shown promising effects on aging markers in animals; the human longevity data so far come only from uncontrolled and observational studies, and the one randomized placebo-controlled trial of Ca-AKG in middle-aged adults has finished enrolling but has not published results. Doses vary by form and purpose, so product labeling is the guide. As a natural metabolic compound, AKG is generally well tolerated, though long-term human data for its longevity use is still developing, and those who are pregnant or on medication should check with a doctor.

Studied Dose Ca-AKG 1,000 mg/day sustained-release is the dose used in longevity products and the ongoing trial. The only completed randomized bone trial used 6 g/day of AKG as the calcium salt.
Active Compound Alpha-ketoglutarate (alpha-KG, 2-oxoglutarate), a TCA cycle intermediate. Forms: calcium AKG (Ca-AKG, most stable), ammonium AKG, sodium AKG.

Benefits

Biological age markers in an uncontrolled study

A longitudinal observational study followed 42 self-reported healthy individuals taking Rejuvant (sustained-release Ca-AKG + sex-specific vitamins) for 4-10 months and reported an average 8-year drop in a DNA methylation age estimate over 7 months. DNA methylation clocks are research tools, not validated clinical endpoints, so a change in a clock reading is not the same as a change in health, function or lifespan. Critical caveats: self-reported, no placebo control, single methylation clock, possible selection bias, small sample, and Ca-AKG combined with vitamins (cannot attribute to AKG alone). Hypothesis-generating, not confirmatory. A later cross-sectional analysis of 4,260 people who bought saliva epigenetic tests found the same delayed-release Ca-AKG plus vitamin product associated with a 1.8-year lower age residual, which is far smaller than 8 years, while plain AKG showed no significant association at all. That analysis is also uncontrolled and open to healthy-user bias.

Randomized trial of Ca-AKG has not reported yet

The Able trial (National University of Singapore Phase 2 RCT) is testing Ca-AKG vs placebo for 6 months in 120 middle-aged adults (40-60 years) with biological age higher than chronological age. Its primary outcome is change in DNA methylation age. Recruitment is finished and all 120 participants were enrolled, and the registry gives a primary completion date of August 2025, but as of August 2026 no results have been published and none are posted on the trial registry, which still lists the study as active and not recruiting with completion estimated for January 2027. Until those results appear this is a study in progress, not a benefit of taking AKG, and the biological age question should be treated as open.

Animal lifespan extension across multiple species

AKG extends lifespan in fruit flies, C. elegans roundworms, and mice. A mouse study showed Ca-AKG reduced frailty and enhanced longevity (compression of morbidity). Mechanism: caloric restriction mimetic via inhibiting ATP synthase and TOR, activating AMPK. Foundational preclinical evidence supporting human longevity research interest. Worth saying plainly: no comparable lifespan or healthspan result has been shown in people, and lifespan extension in short-lived laboratory species has a poor record of carrying over to humans.

Bone density and strength support

Animal studies and one human trial have tested whether Ca-AKG supports bone. The human result landed on bone turnover rather than on bone density. Mechanism: stimulates collagen synthesis (proline hydroxylation requires AKG cofactor) and provides calcium for mineralization. The specific evidence is one randomized double-blind 6-month trial in 76 postmenopausal women with osteopenia, comparing calcium AKG supplying 6 g of AKG per day against the same amount of calcium alone. The bone resorption marker CTX fell by up to 37 percent in the AKG group, with a significant difference from the calcium-only group at 12 and 24 weeks. Because the comparator was calcium alone, that change is attributable to the AKG and not to the calcium it carries. Three limits belong alongside it: osteocalcin did not change, the between-group difference in lumbar spine bone mineral density was 0.9 percent and not statistically significant, and the dose was six times what a typical 1 g Ca-AKG longevity product supplies.

Wound healing and protein synthesis

Older clinical research tested ornithine alpha-ketoglutarate, a different compound from the calcium AKG sold as a supplement, and showed it improves nitrogen balance in surgical patients and burn victims. In severe burn patients it shortened wound healing time and reduced markers of protein breakdown. Mechanism via amino acid synthesis support and growth hormone secretion. Clinical use in some European hospitals as nutritional adjunct. Read this as borrowed evidence rather than a claim for a consumer product. The compound is ornithine AKG, not calcium AKG; the dose was 10 to 30 g per day; it was delivered by feeding tube as part of hospital nutrition; and the patients had burns over a quarter or more of their body surface. None of it has been tested in healthy people taking 1 g of Ca-AKG by mouth.

Muscle protein synthesis support (preclinical)

AKG provides nitrogen carriers for amino acid synthesis (transamination reactions), supporting muscle protein synthesis and reducing protein catabolism in stress states. Animal evidence supports anabolic effects, and the human tests point in both directions. Single-dose trials of arginine alpha-ketoglutarate found nothing: one in resistance-trained and untrained men showed no gain in one-repetition maximum or total load volume on bench or leg press, a second found no improvement in muscular endurance with participants completing slightly fewer chin-ups and total repetitions on the supplement than on placebo, and a third found no added blood flow or nitric oxide response after resistance exercise beyond what the exercise itself produced. One longer study is positive: 12 g/day of arginine alpha-ketoglutarate over 8 weeks of resistance training in 35 men aged 30 to 50 improved bench press one-repetition maximum and peak anaerobic power, with no change in body composition, quadriceps endurance or aerobic capacity. All of these used the arginine salt rather than calcium AKG, the positive trial was small, and its gains were limited to two of the many measures taken, so the fair summary is that a muscle benefit from oral AKG in healthy people is unsettled rather than established.

Mechanism of action

1

TCA cycle intermediate (energy metabolism)

AKG is one of eight TCA cycle intermediates — converted to succinyl-CoA via α-ketoglutarate dehydrogenase. Critical for glucose, fatty acid, and amino acid oxidation. Energy production substrate. Provides direct metabolic support for cellular energy demands.

2

Substrate for dioxygenases (epigenetic regulation)

AKG is a required cofactor for 2-OG-dependent dioxygenases, including TET enzymes (DNA demethylation), JmjC histone demethylases (chromatin modification), prolyl hydroxylases (collagen synthesis, HIF regulation), and many others. Supplementation may support epigenetic regulation, a proposed mechanism for the observed biological age effects.

3

Caloric restriction mimetic via ATP synthase / TOR / AMPK

Animal studies show AKG inhibits ATP synthase and TOR (target of rapamycin) signaling while activating AMPK pathway — mimicking effects of caloric restriction (the most reliable known longevity intervention in animals). Mechanism for lifespan extension observed in flies, worms, mice.

4

Glutamate-glutamine cycling and nitrogen metabolism

AKG combines with ammonia via glutamate dehydrogenase to form glutamate — central nitrogen disposal pathway. Used clinically (post-surgery) to manage nitrogen balance and support amino acid synthesis. Mechanism for protein-anabolic effects in catabolic states.

5

Calcium delivery (Ca-AKG specifically)

Ca-AKG salt provides both alpha-ketoglutarate and calcium — useful for bone health and as practical delivery mechanism. Calcium AKG enhances oral stability and bioavailability vs free AKG. The one human bone trial separated the two components: it compared calcium AKG against an equal amount of calcium alone, so the fall in bone turnover it reported is attributable to the AKG rather than to the calcium the salt carries. Bone mineral density itself did not differ significantly between the two groups, so the calcium delivery is better described as a practical feature of the salt than as a proven bone density benefit.

Clinical trials

1
Rejuvant (Ca-AKG) Biological Age

Longitudinal observational study (Demidenko O, Barardo D, Budovskii V, Finnemore R, Palmer FR 3rd, Kennedy BK, Budovskaya YV 2021, Aging 13(22):24485-24499, doi:10.18632/aging.203736).

42 self-reported healthy individuals taking Rejuvant (sustained-release Ca-AKG + sex-specific vitamins) for 4-10 months. Biological age measured by TruAge DNA methylation test (Horvath-derived clock) before/during/after treatment.

Average 8-YEAR reduction in biological age (TruAge DNA methylation) over average 7 months Rejuvant supplementation. Substantial effect if real. Critical caveats: (1) observational/uncontrolled design, no placebo, (2) self-reported subjects with potential selection bias, (3) single DNA methylation clock, (4) Rejuvant is combination product (AKG + vitamins), (5) sponsored by Ponce de Leon Health (commercial interest), (6) small sample. Most-cited human evidence for AKG biological age effects but methodologically limited.

2
Asadi — Ca-AKG in Mice (Foundational Animal)

Mouse longevity study (Asadi Shahmirzadi A, Edgar D, Liao CY, Hsu YM, Lucanic M, Asadi Shahmirzadi A, Wiley CD, Gan G, Kim DE, Kasler HG, Kuehnemann C, Kaplowitz B, Bhaumik D, Riley RR, Kennedy BK, Lithgow GJ 2020, Cell Metab 32(3):447-456.e6, doi:10.1016/j.cmet.2020.08.004).

C57BL/6 mice received Ca-AKG supplementation. Frailty, lifespan, and healthspan measured.

Ca-AKG reduced frailty and enhanced longevity in mice — compression of morbidity (mice lived longer and with less age-related decline). The mechanism the authors propose is that dietary AKG induces the anti-inflammatory cytokine IL-10, which then suppresses chronic inflammation. Note the direction: IL-10 went up, not down. Several of the investigators disclose equity in the company that sells the Ca-AKG longevity product. Foundational animal evidence supporting Ca-AKG's emergence as 'longevity supplement.' Critical mouse-to-human translation gap — animal lifespan studies do not reliably predict human supplementation effects.

3
ABLE Trial, Phase 2 Ca-AKG vs Placebo, No Results Published

Phase 2 randomized double-blind placebo-controlled trial (NCT05706389). National University of Singapore.

120 healthy middle-aged adults (40-60 years) with biological age higher than chronological age. Randomized to Ca-AKG or placebo for 6 months. Primary outcome: biological age change.

No results. All 120 participants were enrolled and the registry gives a primary completion date of August 2025, but as of August 2026 no results paper has appeared and no results are posted on the registry, which still lists the study as active and not recruiting with completion estimated for January 2027. The only published output so far is a recruitment feasibility report. This entry therefore describes a study design, not a finding, and nothing in it should be read as evidence that Ca-AKG lowers biological age. One correction to the earlier framing: the trial is not fully independent of commercial interest, since one of its investigators has served on the scientific advisory board of the company selling the Ca-AKG product.

Side effects and drug interactions

Common Potential side effects

Generally well-tolerated. The 6 g/day figure comes from a controlled trial in which postmenopausal women took that amount of AKG as the calcium salt for 6 months; that report does not describe adverse effects, though tolerability was not what it set out to measure. Typical consumer doses are far below 6 g.
Mild GI upset (nausea, abdominal discomfort) at high doses.
Allergic reactions: rare.
Pregnancy/lactation: insufficient data.
Long-term safety beyond 12 months: limited data.
Calcium AKG: calcium is roughly 20 percent of the salt by weight, so about 200 mg of elemental calcium per gram. This matters for anyone with hypercalcemia, a history of kidney stones, or an already high total calcium intake from diet and other supplements.

Important Drug interactions

Calcium-containing forms: may interact with bisphosphonates, levothyroxine, fluoroquinolones — separate by 4 hours.
Iron supplements: calcium content of Ca-AKG may reduce non-heme iron absorption; separate by 1-2 hours.
No specific drug interactions have been documented, though that reflects how little AKG has been studied in people rather than a demonstrated clean interaction profile.
Combination use with other supplements has not been tested for safety in any systematic way, so compatibility with other products is assumed rather than demonstrated.
Theoretical: substrates of AKG-dependent dioxygenases (TET, JmjC) — clinical relevance unclear.

Frequently asked questions about Alpha-Ketoglutarate (AKG / Calcium AKG)

What is alpha-ketoglutarate (AKG) used for?

Alpha-ketoglutarate (AKG) is a compound central to cellular energy (the Krebs cycle) and amino acid metabolism. It is used for exercise and recovery, and a form called Ca-AKG is studied in longevity research for healthy aging.

What is AKG good for?

It is used by athletes for performance and recovery (sometimes as arginine-AKG for pumps), though the human trials are mixed: single-dose studies in trained and untrained men found no gain in strength or muscular endurance, while one 8-week training study found a gain in bench press strength and peak power. It is also of growing interest in longevity research, where calcium-AKG has shown promising effects on aging markers in animals. The human longevity evidence is early and comes from uncontrolled studies.

How much alpha-ketoglutarate should I take?

Doses vary by form and purpose; follow product labeling. Longevity-focused calcium-AKG products provide a set daily amount, while sports forms (like arginine-AKG) differ.

Is alpha-ketoglutarate safe?

It is generally well tolerated, as it is a natural metabolic compound. Long-term human data for its longevity use is still developing. As with any supplement, those who are pregnant or on medication should check with a doctor.

What is Alpha-Ketoglutarate?

Alpha-ketoglutarate (AKG) is a compound central to the body's energy-producing Krebs cycle and to amino acid metabolism. It is used by athletes for performance and recovery, sometimes as arginine-AKG for blood-flow support, though the human trials are mixed: single-dose trials in trained and untrained men found no gain…

What is Alpha-Ketoglutarate used for?

Alpha-Ketoglutarate is researched primarily for Longevity, Bone Health, and Muscle & Recovery. A longitudinal observational study followed 42 self-reported healthy individuals taking Rejuvant (sustained-release Ca-AKG + sex-specific vitamins) for 4-10 months and reported an average 8-year drop in a DNA methylation age estimate over 7…

What is the recommended dosage of Alpha-Ketoglutarate?

The clinically studied dose is Ca-AKG 1,000 mg/day sustained-release is the dose used in longevity products and the ongoing trial. The only completed randomized bone trial used 6 g/day of AKG as the calcium salt. Always follow the product label and check with a healthcare provider for personal advice.

Is Alpha-Ketoglutarate safe, and does it have side effects?

For most healthy adults, Alpha-Ketoglutarate is well tolerated at studied doses. Reported effects can include: Generally well-tolerated. The 6 g/day figure comes from a controlled trial in which postmenopausal women took that amount of AKG as the calcium salt for 6 months; that report does not describe adverse effects, though tolerability was not what it set out to measure. It may also interact with some medications. Alpha-Ketoglutarate is not right for everyone, so check with a healthcare provider first if you are pregnant or breastfeeding, have a medical condition, or take prescription medication.

Does Alpha-Ketoglutarate interact with any medications?

Possible interactions include: Calcium-containing forms: may interact with bisphosphonates, levothyroxine, fluoroquinolones — separate by 4 hours. Iron supplements: calcium content of Ca-AKG may reduce non-heme iron absorption; separate by 1-2 hours. If you take prescription medication, check with a pharmacist or doctor before using it.

How strong is the scientific evidence for Alpha-Ketoglutarate?

NutraSmarts rates the evidence for Alpha-Ketoglutarate as Limited (2 out of 5). It is backed by 3 clinical trials and 14 cited references summarized on this page. A higher rating reflects more, larger, and better-designed human studies.

References(14 citations)

Evidence ratings on NutraSmarts are based on the totality of human clinical research, with emphasis on randomized controlled trials, meta-analyses, and systematic reviews. The references below directly support claims made throughout this page.

  1. Demidenko O, Barardo D, Budovskii V, Finnemore R, Palmer FR, Kennedy BK, Budovskaya YV Rejuvant®, a potential life-extending compound formulation with alpha-ketoglutarate and vitamins, conferred an average 8 year reduction in biological aging, after an average of 7 months of use, in the TruAge DNA methylation test Aging (Albany NY). 2021;13(22):24485-24499. doi:10.18632/aging.203736.PubMedUsed to support: Retrospective, uncontrolled analysis of DNA methylation age in 42 people who had bought and taken a calcium alpha-ketoglutarate plus vitamins formulation for an average of 7 months, reporting an average 8-year fall in the methylation age estimate. This is the most cited human result for AKG and biological age, and it is also the weakest form of human evidence: no placebo group, no randomization, self-selected customers, a single methylation clock, and a combination product in which the AKG cannot be separated from the vitamins. The authors include employees and advisors of the companies that sell the supplement and the test. It is the source for the biological age discussion in the benefits section, where the same limits are stated.
  2. Chin RM, Fu X, Pai MY, Vergnes L, Hwang H, Deng G, Diep S, Lomenick B, Meli VS, Monsalve GC, Hu E, Whelan SA, Wang JX, Jung G, Solis GM, Fazlollahi F, Kaweeteerawat C, Quach A, Nili M, Krall AS, Godwin HA, Chang HR, Faull KF, Guo F, Jiang M, Trauger SA, Saghatelian A, Braas D, Christofk HR, Clarke CF, Teitell MA, Petrascheck M, Reue K, Jung ME, Frand AR, Huang J The metabolite α-ketoglutarate extends lifespan by inhibiting ATP synthase and TOR Nature. 2014;510(7505):397-401. doi:10.1038/nature13264.PubMedUsed to support: Laboratory study in the nematode Caenorhabditis elegans showing that alpha-ketoglutarate extends adult worm lifespan by binding and inhibiting ATP synthase, with the effect depending on TOR signaling downstream. This is the origin of the caloric restriction mimetic mechanism described in the mechanisms section. It is a worm study and carries no implication for dose, safety or lifespan in people.
  3. Gyanwali B, Lim ZX, Soh J, Lim C, Guan SP, Goh J, Maier AB, Kennedy BK Alpha-Ketoglutarate dietary supplementation to improve health in humans Trends Endocrinol Metab. 2022;33(2):136-146. doi:10.1016/j.tem.2021.11.003.PubMedUsed to support: Narrative review of AKG supplementation in humans covering biological age, bone, muscle and wound healing. It is useful as an orientation to the field but contains no new data, and its own conclusion is that the human evidence amounts to a few studies from the 1980s and 1990s on muscle growth, wound healing and post-surgical recovery, with no published studies yet showing AKG treating aging or age-related disease. Its senior author is a board member and equity holder in a company that manufactures AKG products.
  4. Sandalova E, Goh J, Lim ZX, Lim ZM, Barardo D, Dorajoo R, Kennedy BK, Maier AB Alpha-ketoglutarate supplementation and BiologicaL agE in middle-aged adults (ABLE)-intervention study protocol Geroscience. 2023;45(5):2897-2907. doi:10.1007/s11357-023-00813-6.PubMedUsed to support: Study protocol only, describing the design of a double-blind placebo-controlled trial of 1 g sustained-release calcium AKG against placebo for 6 months, with 3 months of follow-up, in 120 healthy adults aged 40 to 60 whose DNA methylation age exceeds their chronological age. A protocol reports no findings. It establishes the dose and the design and nothing else, and as of August 2026 the trial's results have not been published or posted. One of the investigators discloses having served on the scientific advisory board of a company selling AKG.
  5. Filip RS, Pierzynowski SG, Lindegard B, et al. Alpha-ketoglutarate decreases serum levels of C-terminal cross-linking telopeptide of type I collagen (CTX) in postmenopausal women with osteopenia: six-month study. Int J Vitam Nutr Res. 2007;77(2):89-97..PubMedUsed to support: Randomized, double-blind, 6-month trial in 76 postmenopausal women with osteopenia, comparing calcium alpha-ketoglutarate supplying 6 g of AKG plus 1.68 g of calcium per day against the same 1.68 g of calcium alone. The bone resorption marker CTX fell by up to 37 percent in the AKG group, with a statistically significant difference from the calcium-only group at 12 and 24 weeks. Because the comparator was calcium alone, the effect is attributable to the AKG rather than to the calcium the salt carries. The limits matter as much as the result: osteocalcin did not change, the between-group difference in lumbar spine bone mineral density was 0.9 percent and not statistically significant, the trial was small, and the dose was six times what a typical 1 g calcium AKG longevity product supplies. This is the completed randomized human trial behind the bone claims in the benefits section, and it is the only trial of its kind for this ingredient.
  6. Asadi Shahmirzadi A, Edgar D, Liao CY, et al. Alpha-Ketoglutarate, an Endogenous Metabolite, Extends Lifespan and Compresses Morbidity in Aging Mice. Cell Metab. 2020;32(3):447-456.e6..PubMedUsed to support: Mouse study feeding calcium alpha-ketoglutarate to C57BL/6 mice, reporting reduced frailty and extended lifespan, described by the authors as a compression of morbidity, with lower systemic inflammatory cytokines and induction of the anti-inflammatory cytokine IL-10 proposed as the mechanism. This is the animal work the longevity positioning rests on, and it is the source for the mouse study described in the clinical trials section. It is a rodent result with no human equivalent, and several of the investigators disclose equity in the company that sells the calcium AKG longevity product.
  7. Lim ZM, Chew YE, Guan L, et al. Recruitment evaluation of a gerotherapeutic randomized controlled trial testing alpha-ketoglutarate in biologically older, middle-aged adults (ABLE). Exp Gerontol. 2025;209:112867..PubMedUsed to support: Recruitment and feasibility report from the randomized placebo-controlled trial of 1 g sustained-release calcium alpha-ketoglutarate against placebo for 6 months in 120 generally healthy adults aged 40 to 60 whose DNA methylation age exceeds their chronological age. It confirms that all 120 participants were enrolled, from 467 who expressed interest. It reports on recruitment only and contains no efficacy result of any kind. Cited in the benefits and clinical trial sections to show that the trial exists and has completed enrolment but has not reported its outcome, which as of August 2026 remains unpublished.
  8. Wax B, Kavazis AN, Webb HE, et al. Acute L-arginine alpha ketoglutarate supplementation fails to improve muscular performance in resistance trained and untrained men. J Int Soc Sports Nutr. 2012;9(1):17..PubMedUsed to support: Randomized, double-blind crossover trial in 8 resistance-trained and 8 untrained men taking 3,000 mg of arginine alpha-ketoglutarate or placebo 45 minutes before exercise. Neither one-repetition maximum nor total load volume on the barbell bench press or leg press differed between supplement and placebo in either group, and heart rate responses were similar. A null result in exactly the population that buys AKG for training, and one reason the muscle and performance discussion in the benefits section is written cautiously. Two qualifications: the form tested was the arginine salt rather than the calcium salt sold for longevity, and the design was an acute single dose rather than a training study.
  9. Greer BK, Jones BT Acute arginine supplementation fails to improve muscle endurance or affect blood pressure responses to resistance training. J Strength Cond Res. 2011;25(7):1789-94..PubMedUsed to support: Crossover trial in 12 trained college-aged men given a serving of arginine alpha-ketoglutarate providing 3,700 mg, or placebo, at two time points, 4 hours and again 30 minutes before exercise, then performing sets of chin-ups, reverse chin-ups and push-ups to exhaustion. Muscular endurance did not improve and blood pressure responses were unaffected; participants completed slightly fewer chin-ups and fewer total repetitions on the supplement than on placebo, and the authors concluded that pre-workout use of these products should be questioned. Small, acute, and using the arginine salt rather than calcium AKG, but it is direct human evidence against the ergogenic claim and it is why the benefits section presents the performance question as unsettled.
  10. Coudray-Lucas C, Le Bever H, Cynober L, et al. Ornithine alpha-ketoglutarate improves wound healing in severe burn patients: a prospective randomized double-blind trial versus isonitrogenous controls. Crit Care Med. 2000;28(6):1772-6..PubMedUsed to support: Prospective, double-blind, randomized trial in 47 patients with burns covering 25 to 95 percent of body surface, given 20 g per day of ornithine alpha-ketoglutarate or an isonitrogenous soy protein control by feeding tube for 3 weeks. Wound healing time was 60 days with ornithine AKG against 90 days with the control for comparable grafted areas, and protein breakdown markers fell in the less severely injured patients. This is the trial behind the wound healing and protein sparing statements in the benefits section, and it is borrowed evidence on several counts at once: the compound is ornithine alpha-ketoglutarate rather than the calcium AKG sold as a supplement, the dose is 20 g per day, delivery was hospital tube feeding rather than swallowing a capsule, and the patients were critically injured rather than healthy.
  11. Pabis K, Wang W, Selvarajoo K, et al. Supplements and Drugs Are Associated With Biological Age in a Cohort of Exceptionally Healthy Individuals. Aging Cell. 2026;25(6):e70517..PubMedUsed to support: Cross-sectional analysis of 4,260 people who bought saliva-based epigenetic age tests between 2020 and 2025 and completed lifestyle and supplement questionnaires, testing 84 commonly used supplements against a biological age residual. A commercially available delayed-release calcium alpha-ketoglutarate plus vitamin product was associated with an average 1.8 years lower age residual, holding up after adjustment for age, sex, smoking and health status, while participants taking plain AKG showed a much smaller and non-significant difference. Important context for the biological age discussion in the benefits section because 1.8 years is roughly a fifth of the 8-year figure from the earlier uncontrolled study of the same product, and because unbranded AKG showed nothing. It remains observational and cross-sectional, with healthy-user and recruitment bias acknowledged by the authors, so it cannot show the supplement caused the difference.
  12. Su Y, Wang T, Wu N, et al. Alpha-ketoglutarate extends Drosophila lifespan by inhibiting mTOR and activating AMPK. Aging (Albany NY). 2019;11(12):4183-4197..PubMedUsed to support: Laboratory study in fruit flies showing that dietary alpha-ketoglutarate extends lifespan, improves climbing ability and heat-stress resistance, and acts by activating AMPK and inhibiting mTOR signaling, alongside a reduced ATP to ADP ratio and increased autophagy. It is the fly component of the cross-species animal lifespan statement in the benefits section, alongside the worm and mouse work. Insect data at micromolar dietary concentrations, carrying no dose, safety or efficacy implication for people, and the supplemented flies also showed reduced reproductive performance.
  13. Campbell B, Roberts M, Kerksick C, et al. Pharmacokinetics, safety, and effects on exercise performance of L-arginine alpha-ketoglutarate in trained adult men. Nutrition. 2006;22(9):872-81..PubMedUsed to support: Randomized, double-blind, placebo-controlled trial in 35 resistance-trained men aged 30 to 50 taking 4 g of arginine alpha-ketoglutarate three times a day, 12 g in total, alongside four days a week of periodized resistance training for 8 weeks. Bench press one-repetition maximum and Wingate peak power improved significantly against placebo, while body composition, total body water, isokinetic quadriceps endurance and aerobic capacity did not. This is the one human trial showing a performance gain from an oral AKG form, and it is why the muscle and recovery claims in the benefits section are kept rather than dropped, but it is also why they are kept cautiously: the form was the arginine salt rather than the calcium AKG sold for longevity, the dose was 12 g a day, the sample was small at 20 supplemented against 15 controls, only two of the many measures taken moved, and shorter single-dose trials of the same salt found nothing.
  14. Willoughby DS, Boucher T, Reid J, et al. Effects of 7 days of arginine-alpha-ketoglutarate supplementation on blood flow, plasma L-arginine, nitric oxide metabolites, and asymmetric dimethyl arginine after resistance exercise. Int J Sport Nutr Exerc Metab. 2011;21(4):291-9..PubMedUsed to support: Randomized trial in 24 physically active men taking 12 g per day of a commercial arginine alpha-ketoglutarate pre-workout product or placebo for 7 days, with brachial artery blood flow, nitric oxide metabolites and hemodynamics measured around a resistance exercise session. Plasma arginine did rise in the supplement group, but blood flow, heart rate, blood pressure and nitric oxide metabolites rose after exercise in both groups with no difference between them, and the authors attributed those changes to the exercise rather than the supplement. This is the direct human test of the blood-flow or pump claim mentioned in the benefits section. It used the arginine salt rather than the calcium AKG sold for longevity, the product tested contained more than one ingredient, and the supplementation period was only 7 days.